Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50009498
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408797BDBM50408797(CHEMBL151228)
Affinity DataKi:  5.50E+3nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 24710BDBM24710(6-chloro-2-methoxyacridin-9-amine | 9-Amino-6-Chlo...)
Affinity DataKi:  7.00E+3nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408796BDBM50408796(CHEMBL153790)
Affinity DataKi:  1.00E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408799BDBM50408799(CHEMBL151397)
Affinity DataKi:  1.10E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50015214BDBM50015214(N-(4-Hydroxy-phenyl)-acetamide | 6-chloro-2-methox...)
Affinity DataKi:  1.90E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084237BDBM50084237([4-(6-Chloro-2-methoxy-acridin-9-ylsulfanyl)-butyl...)
Affinity DataKi:  2.10E+4nMAssay Description:The mixed type inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plots and Cornish-Bowdwn plots.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408798BDBM50408798(CHEMBL152023)
Affinity DataKi:  2.70E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084238BDBM50084238([2-(6-Chloro-2-methoxy-acridin-9-ylsulfanyl)-ethyl...)
Affinity DataKi:  3.70E+4nMAssay Description:The mixed type inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 83820BDBM83820(9-acridin-10-iumamine;chloride | 9-Amino-acridiniu...)
Affinity DataKi:  3.80E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50408800BDBM50408800(TCMDC-141999 | CHEMBL146512)
Affinity DataKi:  4.30E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084237BDBM50084237([4-(6-Chloro-2-methoxy-acridin-9-ylsulfanyl)-butyl...)
Affinity DataKi:  6.70E+4nMAssay Description:The mixed type inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8987BDBM8987(6-chlorotacrine.HCl | CHEMBL486698 | 6-chloro-1,2,...)
Affinity DataKi:  8.00E+4nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50084238BDBM50084238([2-(6-Chloro-2-methoxy-acridin-9-ylsulfanyl)-ethyl...)
Affinity DataKi:  8.30E+4nMAssay Description:The mixed type inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plots and Cornish-Bowdwn plots.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTrypanothione reductase(Trypanosoma cruzi)
Heidelberg University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 8961BDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataKi:  1.40E+5nMAssay Description:The competitive inhibitory activity against trypanothione reductase was evaluated from Lineweaver Burk plotsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed