Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50036897
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Mayo Medical School And Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50369776(CHEMBL298301)
Affinity DataIC50:  2.50E+4nMAssay Description:In vitro inhibition of Farnesyltransferase (FT) by using FT [3H]-SPA kit.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Mayo Medical School And Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50084826(2,5,7-Trinitro-9-oxo-9H-fluorene-4-carboxylic acid...)
Affinity DataIC50:  8.00E+4nMAssay Description:In vitro inhibition of Farnesyltransferase (FT) by using FT [3H]-SPA kit.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Mayo Medical School And Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50084823(2,4,7-Trinitro-5-(piperidine-1-carbonyl)-fluoren-9...)
Affinity DataIC50:  9.60E+4nMAssay Description:In vitro inhibition of Farnesyltransferase (FT) by using FT [3H]-SPA kit.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Mayo Medical School And Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50084824(4-Nitro-2-(2,4,5,7-tetranitro-fluoren-9-ylidenemet...)
Affinity DataIC50:  1.00E+5nMAssay Description:In vitro inhibition of Farnesyltransferase (FT) by using FT [3H]-SPA kit.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
Mayo Medical School And Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50084827(2,7-Dinitro-9-oxo-9H-fluorene-4-carboxylic acid N'...)
Affinity DataIC50:  1.10E+5nMAssay Description:In vitro inhibition of Farnesyltransferase (FT) by using FT [3H]-SPA kit.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed