Affinity DataKi: 5nMAssay Description:Binding affinity against human adenosine A2A receptor using [3H]-CGS-21,680 (95% confidence)More data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against human post-mortem brain adenosine A2A receptor using nuclei caudati and [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity against adenosine A2A receptor of rat brain striatal membranes using [3H]-CGS-21,680More data for this Ligand-Target Pair
Affinity DataKi: 625nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat without and after preincubation with alkaline phosphataseMore data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 1.28E+3nMAssay Description:Binding affinity against adenosine A1 receptor of rat brain cortical membranes using [3H]-CHAMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Binding affinity against human adenosine A1 receptor using [3H]-CCPA (95% confidence)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NECA-induced stimulation of adenylate cyclase at human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of NECA-induced stimulation of adenylate cyclase at human adenosine A2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human adenosine A3 receptor in CHO cell membranes using [3H]-NECAMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against human adenosine A3 receptor in CHO cell membranes using [3H]-NECAMore data for this Ligand-Target Pair