Compile Data Set for Download or QSAR
maximum 50k data
Found 28 Enz. Inhib. hit(s) with all data for entry = 50035080
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085011(2-Benzyloxycarbonylamino-3-(2-{(S)-4-[3-(4,5-dihyd...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085018(3-(2-{(S)-4-[3-(1H-Benzoimidazol-2-ylamino)-propyl...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085015(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(3-guanidino-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085019(2-(3-Benzyl-ureido)-3-{2-[(S)-4-(3-guanidino-propy...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085010(3-{2-[(S)-4-(3-Guanidino-propyl)-2,5-dioxo-imidazo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085006(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(4-guanidino-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085010(3-{2-[(S)-4-(3-Guanidino-propyl)-2,5-dioxo-imidazo...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085008(3-{2-[(S)-4-(3-Guanidino-propyl)-2,5-dioxo-imidazo...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085012(2-(Butane-1-sulfonylamino)-3-{2-[(S)-4-(3-guanidin...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085008(3-{2-[(S)-4-(3-Guanidino-propyl)-2,5-dioxo-imidazo...)
Affinity DataIC50:  550nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085019(2-(3-Benzyl-ureido)-3-{2-[(S)-4-(3-guanidino-propy...)
Affinity DataIC50:  570nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085007(2-Benzyloxycarbonylamino-3-(2-{(S)-4-[N'-(4,5-dihy...)
Affinity DataIC50:  580nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085012(2-(Butane-1-sulfonylamino)-3-{2-[(S)-4-(3-guanidin...)
Affinity DataIC50:  760nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085006(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(4-guanidino-...)
Affinity DataIC50:  850nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085014(2-Benzyloxycarbonylamino-3-(2-{(S)-2,5-dioxo-4-[3-...)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085015(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(3-guanidino-...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085017(2-(3-Benzyl-thioureido)-3-{2-[(S)-4-(3-guanidino-p...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085016(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(2-guanidino-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085013(3-[2-((S)-4-{[(1H-Benzoimidazol-2-ylmethyl)-carbam...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085009(2-Benzyloxycarbonylamino-3-[2-((S)-4-guanidinometh...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085016(2-Benzyloxycarbonylamino-3-{2-[(S)-4-(2-guanidino-...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085014(2-Benzyloxycarbonylamino-3-(2-{(S)-2,5-dioxo-4-[3-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085017(2-(3-Benzyl-thioureido)-3-{2-[(S)-4-(3-guanidino-p...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085007(2-Benzyloxycarbonylamino-3-(2-{(S)-4-[N'-(4,5-dihy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085018(3-(2-{(S)-4-[3-(1H-Benzoimidazol-2-ylamino)-propyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-IIb/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085011(2-Benzyloxycarbonylamino-3-(2-{(S)-4-[3-(4,5-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of fibrinogen binding to integrin alphaIIb-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085013(3-[2-((S)-4-{[(1H-Benzoimidazol-2-ylmethyl)-carbam...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50085009(2-Benzyloxycarbonylamino-3-[2-((S)-4-guanidinometh...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of Kistrin binding to integrin alphaV-beta3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed