Found 17 Enz. Inhib. hit(s) with all data for entry = 50036901 TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.467nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 0.476nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 32.8nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 109nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 152nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 218nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 759nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: 1.07E+3nMAssay Description:Binding affinity was determined by displacement of [3H]- DSLET at Opioid receptor delta 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of [3H]- DAMGO at Opioid receptor mu 1 in rat brain membrane homogenatesMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 165nMAssay Description:Compound was tested for delta antagonist activity against tachykinin NK-1.Tachykinin receptor 1More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 216nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Clinical Research Institute Of Montr£Al
Curated by ChEMBL
Affinity DataIC50: 1.05E+3nMAssay Description:Compound was tested for delta antagonist activity against Tachykinin receptor 1More data for this Ligand-Target Pair
