Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50009583
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085393BDBM50085393((2R,3R)-2-(3-Carbamimidoyl-benzyl)-3-[(3'-carbamoy...)
Affinity DataKi:  0.5nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085402BDBM50085402(4-{4-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allylca...)
Affinity DataKi:  0.75nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085405BDBM50085405(2'-Sulfamoyl-biphenyl-4-carboxylic acid [3-(5-carb...)
Affinity DataKi:  2nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085406BDBM50085406((2R,3R)-3-[(Biphenyl-4-carbonyl)-amino]-2-(3-carba...)
Affinity DataKi:  5nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085390BDBM50085390(Biphenyl-3,4'-dicarboxylic acid 3-amide 4'-{[(E)-3...)
Affinity DataKi:  5nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085392BDBM50085392(Biphenyl-3,4'-dicarboxylic acid 3-amide 4'-{[3-(5-...)
Affinity DataKi:  7nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085388BDBM50085388(3'-Sulfamoyl-biphenyl-4-carboxylic acid [3-(5-carb...)
Affinity DataKi:  9nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085400BDBM50085400(4'-Sulfamoyl-biphenyl-4-carboxylic acid [(E)-3-(5-...)
Affinity DataKi:  12nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085401BDBM50085401(N-[(E)-3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allyl]...)
Affinity DataKi:  19nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085396BDBM50085396(Biphenyl-4,4'-dicarboxylic acid 4-amide 4'-{[3-(5-...)
Affinity DataKi:  20nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085394BDBM50085394(5-Pyridin-2-yl-thiophene-2-carboxylic acid [(E)-3-...)
Affinity DataKi:  37nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085391BDBM50085391(N-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-propyl]-4-...)
Affinity DataKi:  38nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085387BDBM50085387(Biphenyl-4-carboxylic acid [(E)-3-(5-carbamimidoyl...)
Affinity DataKi:  51nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085398BDBM50085398(N-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-propyl]-4-...)
Affinity DataKi:  58nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085395BDBM50085395(4-tert-Butyl-N-[3-(5-carbamimidoyl-2-hydroxy-pheny...)
Affinity DataKi:  59nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085399BDBM50085399(4-tert-Butyl-N-[(E)-3-(5-carbamimidoyl-2-hydroxy-p...)
Affinity DataKi:  61nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085384BDBM50085384(Biphenyl-4-carboxylic acid [3-(5-carbamimidoyl-2-h...)
Affinity DataKi:  88nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085386BDBM50085386(N-[(E)-3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allyl]...)
Affinity DataKi:  128nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085404BDBM50085404(5-Pyridin-2-yl-thiophene-2-carboxylic acid [3-(5-c...)
Affinity DataKi:  131nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085393BDBM50085393((2R,3R)-2-(3-Carbamimidoyl-benzyl)-3-[(3'-carbamoy...)
Affinity DataKi:  140nMAssay Description:Compound was tested for its inhibitory activity against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085403BDBM50085403(6-Chloro-benzo[b]thiophene-2-carboxylic acid [3-(5...)
Affinity DataKi:  181nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085389BDBM50085389(3-Oxo-2,3-dihydro-thieno[3,2-c]pyridazine-6-carbox...)
Affinity DataKi:  184nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085388BDBM50085388(3'-Sulfamoyl-biphenyl-4-carboxylic acid [3-(5-carb...)
Affinity DataKi:  240nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085397BDBM50085397(N-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-propyl]-4-...)
Affinity DataKi:  254nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCoagulation factor X(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085385BDBM50085385(Biphenyl-4-carboxylic acid [3-(3-carbamimidoyl-phe...)
Affinity DataKi:  1.00E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085386BDBM50085386(N-[(E)-3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allyl]...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085394BDBM50085394(5-Pyridin-2-yl-thiophene-2-carboxylic acid [(E)-3-...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085389BDBM50085389(3-Oxo-2,3-dihydro-thieno[3,2-c]pyridazine-6-carbox...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085396BDBM50085396(Biphenyl-4,4'-dicarboxylic acid 4-amide 4'-{[3-(5-...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085405BDBM50085405(2'-Sulfamoyl-biphenyl-4-carboxylic acid [3-(5-carb...)
Affinity DataKi:  1.50E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085400BDBM50085400(4'-Sulfamoyl-biphenyl-4-carboxylic acid [(E)-3-(5-...)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085401BDBM50085401(N-[(E)-3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allyl]...)
Affinity DataKi:  1.80E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085391BDBM50085391(N-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-propyl]-4-...)
Affinity DataKi:  1.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085402BDBM50085402(4-{4-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-allylca...)
Affinity DataKi:  2.20E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085395BDBM50085395(4-tert-Butyl-N-[3-(5-carbamimidoyl-2-hydroxy-pheny...)
Affinity DataKi:  2.20E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085399BDBM50085399(4-tert-Butyl-N-[(E)-3-(5-carbamimidoyl-2-hydroxy-p...)
Affinity DataKi:  2.30E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085404BDBM50085404(5-Pyridin-2-yl-thiophene-2-carboxylic acid [3-(5-c...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085392BDBM50085392(Biphenyl-3,4'-dicarboxylic acid 3-amide 4'-{[3-(5-...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085384BDBM50085384(Biphenyl-4-carboxylic acid [3-(5-carbamimidoyl-2-h...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085387BDBM50085387(Biphenyl-4-carboxylic acid [(E)-3-(5-carbamimidoyl...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085390BDBM50085390(Biphenyl-3,4'-dicarboxylic acid 3-amide 4'-{[(E)-3...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085403BDBM50085403(6-Chloro-benzo[b]thiophene-2-carboxylic acid [3-(5...)
Affinity DataKi: >2.90E+3nMAssay Description:In vitro inhibition of trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085396BDBM50085396(Biphenyl-4,4'-dicarboxylic acid 4-amide 4'-{[3-(5-...)
Affinity DataKi:  2.90E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085399BDBM50085399(4-tert-Butyl-N-[(E)-3-(5-carbamimidoyl-2-hydroxy-p...)
Affinity DataKi:  3.20E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlasminogen(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085392BDBM50085392(Biphenyl-3,4'-dicarboxylic acid 3-amide 4'-{[3-(5-...)
Affinity DataKi:  3.50E+3nMAssay Description:Compound was tested for its inhibitory activity against PlasminMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085405BDBM50085405(2'-Sulfamoyl-biphenyl-4-carboxylic acid [3-(5-carb...)
Affinity DataKi: >4.00E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085391BDBM50085391(N-[3-(5-Carbamimidoyl-2-hydroxy-phenyl)-propyl]-4-...)
Affinity DataKi: >4.00E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085400BDBM50085400(4'-Sulfamoyl-biphenyl-4-carboxylic acid [(E)-3-(5-...)
Affinity DataKi: >4.00E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085389BDBM50085389(3-Oxo-2,3-dihydro-thieno[3,2-c]pyridazine-6-carbox...)
Affinity DataKi: >4.00E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProthrombin(Human)
Rhone-Poulenc Rorer

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085404BDBM50085404(5-Pyridin-2-yl-thiophene-2-carboxylic acid [3-(5-c...)
Affinity DataKi: >4.00E+3nMAssay Description:In vitro inhibition of coagulation factor IIa.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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