Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50036907
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118238BDBM50118238(MRS 2279 | CHEMBL339873)
Affinity DataIC50: 51.6nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085314BDBM50085314(Phosphoric acid mono-[4-(6-methylamino-purin-9-ylm...)
Affinity DataIC50: 148nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085825BDBM50085825(Phosphoric acid mono-[4-(6-amino-purin-9-yl)-1-pho...)
Affinity DataEC50:  155nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085821BDBM50085821(Phosphoric acid mono-[4-(6-methylamino-purin-9-yl)...)
Affinity DataIC50: 157nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085322BDBM50085322(Phosphoric acid mono-[5-(2-chloro-6-methylamino-pu...)
Affinity DataIC50: 206nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118229BDBM50118229(MRS 2179 | CHEMBL129841)
Affinity DataIC50: 331nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085826BDBM50085826(Phosphoric acid mono-[5-(6-methylamino-2-methylsul...)
Affinity DataIC50: 362nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085817BDBM50085817(Phosphoric acid mono-[5-(2-chloro-6-methylamino-pu...)
Affinity DataIC50: 566nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085824BDBM50085824(Phosphoric acid mono-[3-(2-chloro-6-methylamino-pu...)
Affinity DataIC50: 805nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085823BDBM50085823(Phosphoric acid mono-[5-(6-methylamino-purin-9-yl)...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085828BDBM50085828(Phosphoric acid mono-[5-(2-amino-6-methylamino-pur...)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085818BDBM50085818(N6-Methyl-1,5-anhydro-2-(adenin-9-yl)-2,3-dideoxy-...)
Affinity DataIC50: 2.37E+3nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085313BDBM50085313(Phosphoric acid mono-[4-(6-amino-purin-9-ylmethyl)...)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50076474BDBM50076474(Phosphoric acid mono-[5-(6-amino-purin-9-yl)-2-pho...)
Affinity DataEC50:  2.99E+3nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085829BDBM50085829(Phosphoric acid mono-[4-(2-amino-6-methylamino-pur...)
Affinity DataIC50: 5.42E+3nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085829BDBM50085829(Phosphoric acid mono-[4-(2-amino-6-methylamino-pur...)
Affinity DataEC50:  6.51E+3nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085313BDBM50085313(Phosphoric acid mono-[4-(6-amino-purin-9-ylmethyl)...)
Affinity DataEC50:  7.21E+3nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085818BDBM50085818(N6-Methyl-1,5-anhydro-2-(adenin-9-yl)-2,3-dideoxy-...)
Affinity DataEC50:  9.35E+3nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085822BDBM50085822(Phosphoric acid mono-[1-(6-amino-purin-9-yl)-4-pho...)
Affinity DataEC50:  1.89E+4nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085820BDBM50085820({2-[2-(6-Amino-purin-9-yl)-6-phosphonooxymethyl-mo...)
Affinity DataEC50:  3.70E+4nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085822BDBM50085822(Phosphoric acid mono-[1-(6-amino-purin-9-yl)-4-pho...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of 30 nM 2-MeSADP stimulation of 2PY1-mediated phospholipase C (PLC) activity in Turkey erythrocyte ghostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetP2Y purinoceptor 1(Wild turkey)
National Institute of Diabetes

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085827BDBM50085827(Phosphoric acid mono-[5-(6-methylamino-purin-9-yl)...)
Affinity DataEC50:  4.10E+4nMAssay Description:In vitro stimulation of 2PY1 purinoceptor mediated phospholipase C (PLC) activity in Turkey Erythrocyte GhostsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed