Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50009865
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50056378(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088696(3-Amino-6-ethyl-2-{3-[4-(2-methoxy-phenyl)-piperaz...)
Affinity DataKi:  0.190nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088686(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50056384(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  0.650nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088693(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088690(3-Amino-5,6-dimethyl-2-{3-[4-(2-nitro-phenyl)-pipe...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50056384(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088695(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyls...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088692(3-Amino-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-p...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50056362(3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088688(3-Amino-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-pro...)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50056378(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088689(1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088686(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088691(3-Amino-6-ethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088687(3-Amino-6-ethyl-2-{3-[4-(2-nitro-phenyl)-piperazin...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088695(2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyls...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088693(3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088696(3-Amino-6-ethyl-2-{3-[4-(2-methoxy-phenyl)-piperaz...)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088689(1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088692(3-Amino-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-p...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088690(3-Amino-5,6-dimethyl-2-{3-[4-(2-nitro-phenyl)-pipe...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandPNGBDBM50088694(1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...)
Affinity DataKi:  135nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088687(3-Amino-6-ethyl-2-{3-[4-(2-nitro-phenyl)-piperazin...)
Affinity DataKi:  195nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088688(3-Amino-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-pro...)
Affinity DataKi:  366nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50056362(3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...)
Affinity DataKi:  434nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088694(1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...)
Affinity DataKi:  437nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50088691(3-Amino-6-ethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1...)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed