Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50009944
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089314(CHEMBL405182 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...)
Affinity DataKi:  0.0230nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089307(CHEMBL410579 | H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D...)
Affinity DataKi:  0.0350nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089308(CHEMBL412349 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic...)
Affinity DataKi:  0.0800nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...)
Affinity DataKi:  0.110nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089313(CHEMBL412824 | H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-...)
Affinity DataKi:  0.220nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089313(CHEMBL412824 | H-Lys-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT-...)
Affinity DataKi:  0.400nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089310(2-({1-[2-(2-{2-[(1-{1-[2-(2,6-Diamino-hexanoylamin...)
Affinity DataKi:  0.900nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089312(CHEMBL408846 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT...)
Affinity DataKi:  4.40nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089309(CHEMBL216618 | H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT...)
Affinity DataKi:  5.60nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089314(CHEMBL405182 | H-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT-...)
Affinity DataKi:  9.20nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089310(2-({1-[2-(2-{2-[(1-{1-[2-(2,6-Diamino-hexanoylamin...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089308(CHEMBL412349 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-DTic...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50049949((BK) H-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Phe-Arg-OH | (b...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089306(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pentano...)
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089311(CHEMBL385367 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-Ti...)
Affinity DataKi:  24nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089307(CHEMBL410579 | H-Lys-Lys-Arg-Pro-Hyp-Gly-Igl-Ser-D...)
Affinity DataKi:  62nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089312(CHEMBL408846 | H-DArg-Arg-Pro-Hyp-Gly-Thi-Ser-D-BT...)
Affinity DataKi:  83nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089309(CHEMBL216618 | H-DArg-Arg-Pro-Hyp-Gly-Igl-Ser-D-BT...)
Affinity DataKi:  325nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50089306(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pentano...)
Affinity DataKi:  382nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed