Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50010080
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataIC50:  2nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090745(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  7nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090748(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  11nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090736(1-{2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  14nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090732(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  16nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090724(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  17nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090730(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  20nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090734(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  23nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090723(1-{2-[2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  25nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090728(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  28nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090752(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  28nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090725(1-{2-[2-({2-[2-(2-Acetylamino-3-naphthalen-2-yl-pr...)
Affinity DataIC50:  31nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090737(1-[2-(3-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  38nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090727(1-{2-[(1-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pr...)
Affinity DataIC50:  42nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090747(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50:  45nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090744(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50:  70nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090750(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  72nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090739(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  74nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090733(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  81nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090746(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  88nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090738(Ac-D-Nal2-D-Cpa-D-Pal-Pro-Arg-Pro-D-Ala-NH2 | CHEM...)
Affinity DataIC50:  110nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090743(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  130nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090729(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50:  130nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090749(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50:  140nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090751(1-[2-(2-{2-[2-(2-Acetylamino-3-phenyl-propionylami...)
Affinity DataIC50:  230nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090753(1-[2-(2-{2-[2-(2-Amino-3-naphthalen-2-yl-propionyl...)
Affinity DataIC50:  280nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090735(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-1-yl-pro...)
Affinity DataIC50:  370nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090740(1-{2-[2-(2-{2-[2-Acetylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50:  450nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090742(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50:  550nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090726(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50:  1.50E+3nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Institute Of Science

Curated by ChEMBL
LigandPNGBDBM50090741(CHEMBL409979 | [1-(1-{1-[({1-[2-(1-Carbamoyl-ethyl...)
Affinity DataIC50:  2.20E+3nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed