Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50036833
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090943(3-(2-{4-[3-(2-Bromo-6-chloro-phenyl)-5-isopropyl-i...)
Affinity DataEC50:  12nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM21724(3-[(E)-2-(2-chloro-4-{[3-(2,6-dichlorophenyl)-5-(p...)
Affinity DataEC50:  15nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090948(4-(2-{4-[3-(2,6-Dichloro-phenyl)-5-isopropyl-isoxa...)
Affinity DataEC50:  37nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090939(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-isopropyl-isoxa...)
Affinity DataEC50:  47nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090944(3-(2-{2-Chloro-4-[5-ethyl-3-(2-trifluoromethoxy-ph...)
Affinity DataEC50:  48nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090945(3-(2-{2-Chloro-4-[5-ethyl-3-(2-fluoro-6-trifluorom...)
Affinity DataEC50:  54nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090947(3-(2-{2-Chloro-4-[3-(2,6-dichloro-benzyl)-5-ethyl-...)
Affinity DataEC50:  60nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090940(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-methyl-isoxazol...)
Affinity DataEC50:  70nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090942(4-(2-{4-[3-(2,6-Dichloro-phenyl)-5-ethyl-isoxazol-...)
Affinity DataEC50:  100nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM50090941(3-(2-{4-[3-(2,6-Dichloro-phenyl)-5-isopropyl-isoxa...)
Affinity DataEC50:  100nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Glaxo Wellcome Research & Development

Curated by ChEMBL
LigandPNGBDBM21674(Chenodeoxycholic Acid | CDCA | (4R)-4-[(1S,2S,5R,7...)
Affinity DataEC50:  3.40E+3nMAssay Description:Ligand dependent recruitment of SRC1(676-700) peptide to human Farnesoid X-activated receptor by fluorescence resonance energy transfer assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)