Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 593
TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4213(6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4...)
Affinity DataIC50:  8nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4193(1,6-naphthyridin-2(1H)-one deriv. 8r | 3-(2,6-Dich...)
Affinity DataIC50:  11nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4214(4-{[6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7H,8H-py...)
Affinity DataIC50:  14nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4186(1,6-naphthyridin-2(1H)-one deriv. 7s | 3-(2,6-Dich...)
Affinity DataIC50:  16nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4188(1,6-naphthyridin-2(1H)-one deriv. 7u | 3-(2,6-Dich...)
Affinity DataIC50:  23nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4174(1,6-naphthyridin-2(1H)-one deriv. 7g | 3-(2,6-Dich...)
Affinity DataIC50:  24nMpH: 7.5 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4187(1,6-naphthyridin-2(1H)-one deriv. 7t | 3-(2,6-Dich...)
Affinity DataIC50:  28nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4185(1,6-naphthyridin-2(1H)-one deriv. 7r | 3-(2,6-Dich...)
Affinity DataIC50:  32nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4177(1,6-naphthyridin-2(1H)-one deriv. 7j | 3-(2,6-Dich...)
Affinity DataIC50:  35nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4176(1,6-naphthyridin-2(1H)-one deriv. 7i | 3-(2,6-Dich...)
Affinity DataIC50:  41nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4188(1,6-naphthyridin-2(1H)-one deriv. 7u | 3-(2,6-Dich...)
Affinity DataIC50:  42nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4191(1,6-naphthyridin-2(1H)-one deriv. 8f | 3-(2,6-Dich...)
Affinity DataIC50:  42nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4173(1,6-naphthyridin-2(1H)-one deriv. 7f | 3-(2,6-Dich...)
Affinity DataIC50:  44nMpH: 7.5 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4179(1,6-naphthyridin-2(1H)-one deriv. 7l | 3-(2,6-Dich...)
Affinity DataIC50:  45nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4175(1,6-naphthyridin-2(1H)-one deriv. 7h | 3-(2,6-Dich...)
Affinity DataIC50:  59nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4192(1,6-naphthyridin-2(1H)-one deriv. 8h | 3-(2,6-dich...)
Affinity DataIC50:  72nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4184(1,6-naphthyridin-2(1H)-one deriv. 7q | 3-(2,6-Dich...)
Affinity DataIC50:  78nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4173(1,6-naphthyridin-2(1H)-one deriv. 7f | 3-(2,6-Dich...)
Affinity DataIC50:  80nMpH: 7.0 T: 25°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4174(1,6-naphthyridin-2(1H)-one deriv. 7g | 3-(2,6-Dich...)
Affinity DataIC50:  80nMpH: 7.0 T: 25°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4184(1,6-naphthyridin-2(1H)-one deriv. 7q | 3-(2,6-Dich...)
Affinity DataIC50:  100nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4213(6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4...)
Affinity DataIC50:  100nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4192(1,6-naphthyridin-2(1H)-one deriv. 8h | 3-(2,6-dich...)
Affinity DataIC50:  110nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4177(1,6-naphthyridin-2(1H)-one deriv. 7j | 3-(2,6-Dich...)
Affinity DataIC50:  110nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4187(1,6-naphthyridin-2(1H)-one deriv. 7t | 3-(2,6-Dich...)
Affinity DataIC50:  120nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4184(1,6-naphthyridin-2(1H)-one deriv. 7q | 3-(2,6-Dich...)
Affinity DataIC50:  130nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4172(1,6-naphthyridin-2(1H)-one deriv. 7e | 3-(2,6-Dich...)
Affinity DataIC50:  150nMpH: 7.0 T: 25°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4191(1,6-naphthyridin-2(1H)-one deriv. 8f | 3-(2,6-Dich...)
Affinity DataIC50:  170nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4176(1,6-naphthyridin-2(1H)-one deriv. 7i | 3-(2,6-Dich...)
Affinity DataIC50:  170nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4175(1,6-naphthyridin-2(1H)-one deriv. 7h | 3-(2,6-Dich...)
Affinity DataIC50:  170nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4214(4-{[6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7H,8H-py...)
Affinity DataIC50:  180nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4178(1,6-naphthyridin-2(1H)-one deriv. 7k | 3-(2,6-Dich...)
Affinity DataIC50:  200nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4186(1,6-naphthyridin-2(1H)-one deriv. 7s | 3-(2,6-Dich...)
Affinity DataIC50:  210nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4180(1,6-naphthyridin-2(1H)-one deriv. 7m | 3-(2,6-Dich...)
Affinity DataIC50:  210nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4169(1,6-naphthyridin-2(1H)-one deriv. 7b | 3-(2,6-Dich...)
Affinity DataIC50:  210nMpH: 7.0 T: 25°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4179(1,6-naphthyridin-2(1H)-one deriv. 7l | 3-(2,6-Dich...)
Affinity DataIC50:  230nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4189(1,6-naphthyridin-2(1H)-one deriv. 7v | 3-(2,6-Dich...)
Affinity DataIC50:  250nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4185(1,6-naphthyridin-2(1H)-one deriv. 7r | 3-(2,6-Dich...)
Affinity DataIC50:  250nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4186(1,6-naphthyridin-2(1H)-one deriv. 7s | 3-(2,6-Dich...)
Affinity DataIC50:  260nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4188(1,6-naphthyridin-2(1H)-one deriv. 7u | 3-(2,6-Dich...)
Affinity DataIC50:  260nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4214(4-{[6-(2,6-dichlorophenyl)-8-methyl-7-oxo-7H,8H-py...)
Affinity DataIC50:  290nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4172(1,6-naphthyridin-2(1H)-one deriv. 7e | 3-(2,6-Dich...)
Affinity DataIC50:  300nMpH: 7.5 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4168(1,6-naphthyridin-2(1H)-one deriv. 7a | 7-Amino-3-(...)
Affinity DataIC50:  350nMpH: 7.5 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4185(1,6-naphthyridin-2(1H)-one deriv. 7r | 3-(2,6-Dich...)
Affinity DataIC50:  360nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4168(1,6-naphthyridin-2(1H)-one deriv. 7a | 7-Amino-3-(...)
Affinity DataIC50:  380nMpH: 7.0 T: 25°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4169(1,6-naphthyridin-2(1H)-one deriv. 7b | 3-(2,6-Dich...)
Affinity DataIC50:  420nMpH: 7.5 T: 22°CAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4193(1,6-naphthyridin-2(1H)-one deriv. 8r | 3-(2,6-Dich...)
Affinity DataIC50:  440nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4180(1,6-naphthyridin-2(1H)-one deriv. 7m | 3-(2,6-Dich...)
Affinity DataIC50:  540nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProto-oncogene tyrosine-protein kinase Src(Human)
University of Auckland

LigandPNGBDBM4182(1,6-naphthyridin-2(1H)-one deriv. 7o | 3-(2,6-Dich...)
Affinity DataIC50:  550nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetFibroblast growth factor receptor 1(Human)
University of Auckland

LigandPNGBDBM4178(1,6-naphthyridin-2(1H)-one deriv. 7k | 3-(2,6-Dich...)
Affinity DataIC50:  570nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetPlatelet-derived growth factor receptor beta(Human)
University of Auckland

LigandPNGBDBM4213(6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4...)
Affinity DataIC50:  640nMAssay Description:IC50 is the inhibitor concentration which inhibits 50% of kinase activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] labe...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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