Compile Data Set for Download or QSAR
maximum 50k data
Found 115 Enz. Inhib. hit(s) with all data for entry = 50010160
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091652(CHEMBL269503 | PYY | PYY, rat | Peptide YY(PYY)(YP...)
Affinity DataIC50:  0.0200nMAssay Description:Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091672(CHEMBL412704 | N-alpha-Ac-[CH2-NH35-36]PYY(22-36)-...)
Affinity DataIC50:  0.0500nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091652(CHEMBL269503 | PYY | PYY, rat | Peptide YY(PYY)(YP...)
Affinity DataIC50:  0.0700nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091652(CHEMBL269503 | PYY | PYY, rat | Peptide YY(PYY)(YP...)
Affinity DataIC50:  0.140nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091663(CHEMBL214707 | N-alpha-Ac-[Trp30,CH2-NH-35-36]PYY(...)
Affinity DataIC50:  0.280nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091684(CHEMBL412257 | N-alpha-Ac-[Nle24,28,Trp30,Nva31,CH...)
Affinity DataIC50:  0.310nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50005530(CHEMBL267633 | D-Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-G...)
Affinity DataIC50:  0.320nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091669(CHEMBL438923 | N-alpha-Ac-[CH2-NH28-29]PYY(22-36)-...)
Affinity DataIC50:  0.360nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091679(CHEMBL441007 | bis(24/24'){N-alpha-Ac-[Cys24]PYY(2...)
Affinity DataIC50:  0.390nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091651(CHEMBL411200 | N-alpha-Ac-[Nle24,28,Trp30,Nva31]PY...)
Affinity DataIC50:  0.560nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091653(CHEMBL266021 | N-alpha-Ac-[Nle24,28,30,Nva31]PYY(2...)
Affinity DataIC50:  0.590nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091661(CHEMBL410938 | N-alpha-Ac-[Trp28]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  0.600nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091674(CHEMBL412698 | N-alpha-Ac-[D-Trp30]PYY(22-36)-NH2(...)
Affinity DataIC50:  0.600nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091679(CHEMBL441007 | bis(24/24'){N-alpha-Ac-[Cys24]PYY(2...)
Affinity DataIC50:  0.630nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091668(AcPYY(22-36) | CHEMBL269267 | N-alpha-Ac-PYY(22-36...)
Affinity DataIC50:  0.910nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091674(CHEMBL412698 | N-alpha-Ac-[D-Trp30]PYY(22-36)-NH2(...)
Affinity DataIC50:  0.980nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091650(Ala-Ser-Leu-Arg-His-Thi-Leu-Asn-Leu-Val-Thr-Arg-Gl...)
Affinity DataIC50:  1nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091659(CHEMBL384306 | N-alpha-Ac-[Trp27,CH2-NH-35-36]PYY(...)
Affinity DataIC50:  1.05nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091685(CHEMBL411637 | N-alpha-Ac-[Trp28,30]PYY(22-36)-NH2...)
Affinity DataIC50:  1.07nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091662(CHEMBL410792 | N-alpha-Ac-[Nal30]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  1.09nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091659(CHEMBL384306 | N-alpha-Ac-[Trp27,CH2-NH-35-36]PYY(...)
Affinity DataIC50:  1.12nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091676(CHEMBL429905 | N-alpha-Ac-[Phe27,36]PYY(22-36)-NH2...)
Affinity DataIC50:  1.16nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091668(AcPYY(22-36) | CHEMBL269267 | N-alpha-Ac-PYY(22-36...)
Affinity DataIC50:  1.30nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091672(CHEMBL412704 | N-alpha-Ac-[CH2-NH35-36]PYY(22-36)-...)
Affinity DataIC50:  1.32nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091663(CHEMBL214707 | N-alpha-Ac-[Trp30,CH2-NH-35-36]PYY(...)
Affinity DataIC50:  1.39nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091684(CHEMBL412257 | N-alpha-Ac-[Nle24,28,Trp30,Nva31,CH...)
Affinity DataIC50:  1.75nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091666(CHEMBL413612 | N-alpha-Ac-[Phe27]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  1.83nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50005530(CHEMBL267633 | D-Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-G...)
Affinity DataIC50:  2nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091661(CHEMBL410938 | N-alpha-Ac-[Trp28]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  2.08nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091670(CHEMBL428320 | N-alpha-Ac-[Trp27]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  2.09nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091683(CHEMBL438096 | N-alpha-Ac-[Trp24]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  2.10nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091666(CHEMBL413612 | N-alpha-Ac-[Phe27]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  2.30nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091675(CHEMBL412378 | N-alpha-Ac-[Bip27]PYY(22-36)-NH2)
Affinity DataIC50:  2.42nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091650(Ala-Ser-Leu-Arg-His-Thi-Leu-Asn-Leu-Val-Thr-Arg-Gl...)
Affinity DataIC50:  2.63nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091658(CHEMBL427594 | N-alpha-Ac-[Tyr22,Phe27]PYY(22-36)-...)
Affinity DataIC50:  2.68nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091655(CHEMBL438411 | [Leu31, Pro34]PYY(YPAKPEAPGEDASPEEL...)
Affinity DataIC50:  2.69nMAssay Description:Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091667(CHEMBL428292 | N-alpha-Ac-[CH2-NH24-25]PYY(22-36)-...)
Affinity DataIC50:  2.76nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50005530(CHEMBL267633 | D-Tyr-Pro-Ser-Lys-Pro-Asp-Asn-Pro-G...)
Affinity DataIC50:  3.07nMAssay Description:Affinity against Neuropeptide Y receptor Y1 in SK-N-MC cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091685(CHEMBL411637 | N-alpha-Ac-[Trp28,30]PYY(22-36)-NH2...)
Affinity DataIC50:  3.17nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091670(CHEMBL428320 | N-alpha-Ac-[Trp27]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  3.20nMAssay Description:Tested for the affinity for intestinal PYY from rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091658(CHEMBL427594 | N-alpha-Ac-[Tyr22,Phe27]PYY(22-36)-...)
Affinity DataIC50:  3.40nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091687(CHEMBL263350 | N-alpha-Ac-[Tic27]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  3.40nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091662(CHEMBL410792 | N-alpha-Ac-[Nal30]PYY(22-36)-NH2(N-...)
Affinity DataIC50:  3.54nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091651(CHEMBL411200 | N-alpha-Ac-[Nle24,28,Trp30,Nva31]PY...)
Affinity DataIC50:  3.73nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091671(CHEMBL425095 | N-alpha-Ac-[Ala26,Phe27]PYY(22-36)-...)
Affinity DataIC50:  3.84nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091681(CHEMBL406128 | N-alpha-Ac-[CH2-NH25-26]PYY(22-36)-...)
Affinity DataIC50:  4.22nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091678(Ala-Ser-Leu-Arg-His-Phe-Leu-Asn-Leu-Val-Thr-Arg-Gl...)
Affinity DataIC50:  4.5nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091680(CHEMBL411800 | N-alpha-Ac-[CH2-NH32-33]PYY(22-36)-...)
Affinity DataIC50:  5.03nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091671(CHEMBL425095 | N-alpha-Ac-[Ala26,Phe27]PYY(22-36)-...)
Affinity DataIC50:  5.30nMAssay Description:Antisecretory potency, affinity for intestinal PYY of rat jejunum by using short circuit current (SCC) method.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(Homo sapiens (Human))
University Of Cincinnati Medical Center

Curated by ChEMBL
LigandPNGBDBM50091677(CHEMBL405527 | N-alpha-Ac-[Phe22,27]PYY(22-36)-NH2...)
Affinity DataIC50:  5.61nMAssay Description:Affinity against Neuropeptide Y receptor Y2 in SK-N-BE2 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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