Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 50003559
TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50005463BDBM50005463(1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-phen...)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81962BDBM81962(S-L-365,260)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Rat)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50449787BDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataKi:  0.148nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type A receptor of rat pancreatic membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472889BDBM50472889(CHEMBL415240)
Affinity DataKi:  0.178nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472863BDBM50472863(CHEMBL333979)
Affinity DataKi:  0.209nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472878BDBM50472878(CHEMBL331872)
Affinity DataKi:  0.224nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472863BDBM50472863(CHEMBL333979)
Affinity DataKi:  0.251nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472898BDBM50472898(CHEMBL332902)
Affinity DataKi:  0.288nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472855BDBM50472855(CHEMBL331468)
Affinity DataKi:  0.295nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472870BDBM50472870(CHEMBL331975)
Affinity DataKi:  0.302nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472884BDBM50472884(CHEMBL121021)
Affinity DataKi:  0.331nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50449787BDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataKi:  0.355nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472854BDBM50472854(CHEMBL330977)
Affinity DataKi:  0.372nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472887BDBM50472887(CHEMBL330773)
Affinity DataKi:  0.490nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472864BDBM50472864(CHEMBL402702)
Affinity DataKi:  0.562nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472853BDBM50472853(CHEMBL331244)
Affinity DataKi:  0.575nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472876BDBM50472876(CHEMBL332568)
Affinity DataKi:  0.603nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472885BDBM50472885(CHEMBL118622)
Affinity DataKi:  0.646nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472871BDBM50472871(CHEMBL118954)
Affinity DataKi:  0.661nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472886BDBM50472886(CHEMBL421271)
Affinity DataKi:  0.676nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472848BDBM50472848(CHEMBL420728)
Affinity DataKi:  0.676nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472851BDBM50472851(CHEMBL331763)
Affinity DataKi:  0.676nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472854BDBM50472854(CHEMBL330977)
Affinity DataKi:  0.708nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type B receptor of guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472895BDBM50472895(CHEMBL120296)
Affinity DataKi:  0.724nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472882BDBM50472882(CHEMBL332403)
Affinity DataKi:  0.724nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472847BDBM50472847(CHEMBL121331)
Affinity DataKi:  0.759nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472857BDBM50472857(CHEMBL121028)
Affinity DataKi:  0.832nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472854BDBM50472854(CHEMBL330977)
Affinity DataKi:  0.933nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472865BDBM50472865(CHEMBL331971)
Affinity DataKi:  0.955nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472893BDBM50472893(CHEMBL333517)
Affinity DataKi:  0.955nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472873BDBM50472873(CHEMBL120363)
Affinity DataKi:  0.977nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472892BDBM50472892(CHEMBL331262)
Affinity DataKi:  1nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472866BDBM50472866(CHEMBL120021)
Affinity DataKi:  1.10nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472890BDBM50472890(CHEMBL339879)
Affinity DataKi:  1.10nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472875BDBM50472875(CHEMBL333930)
Affinity DataKi:  1.30nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472851BDBM50472851(CHEMBL331763)
Affinity DataKi:  1.30nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472900BDBM50472900(CHEMBL331119)
Affinity DataKi:  1.30nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472874BDBM50472874(CHEMBL118189)
Affinity DataKi:  1.40nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50211670BDBM50211670(CHEMBL103750)
Affinity DataKi:  1.5nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472880BDBM50472880(CHEMBL338278)
Affinity DataKi:  1.5nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472859BDBM50472859(CHEMBL120031)
Affinity DataKi:  1.5nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472850BDBM50472850(CHEMBL278018)
Affinity DataKi:  1.5nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 81962BDBM81962(S-L-365,260)
Affinity DataKi:  1.60nMAssay Description:Inhibition by displacing [3H]CCK-8S against human Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472861BDBM50472861(CHEMBL121267)
Affinity DataKi:  1.70nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472869BDBM50472869(CHEMBL331405)
Affinity DataKi:  1.90nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472863BDBM50472863(CHEMBL333979)
Affinity DataKi:  1.90nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472891BDBM50472891(CHEMBL334020)
Affinity DataKi:  1.90nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50449787BDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataKi:  1.90nMAssay Description:Inhibition by displacing [3H]CCK-8S against Cholecystokinin type B receptor of guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472862BDBM50472862(CHEMBL332595)
Affinity DataKi:  2.10nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Glaxo Wellcome Medicines Research Centre

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472896BDBM50472896(CHEMBL331688)
Affinity DataKi:  2.10nMAssay Description:In vitro inhibition of binding of [3H]pCCK-8 against Cholecystokinin type B receptor of guinea pig cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 142 total ) | Next | Last >>
Jump to: