Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50010307
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093113(CHEMBL306097 | N-{1-[2-(4-{5-(3,5-Bis-trifluoromet...)
Affinity DataKi:  9nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093118(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093104(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093107(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  13nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093120(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093111(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093107(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  14nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093105(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  16nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093097(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093102(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093120(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093086(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093116(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  22nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093112(5-[4-(2-Azetidin-1-yl-2-oxo-ethyl)-piperazin-1-yl]...)
Affinity DataKi:  23nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093110((S)-1-[2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)...)
Affinity DataKi:  24nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093123(1-[2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(...)
Affinity DataKi:  24nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093104(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  24nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093086(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  25nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093110((S)-1-[2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093097(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093105(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093124(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  30nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093116(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  31nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093112(5-[4-(2-Azetidin-1-yl-2-oxo-ethyl)-piperazin-1-yl]...)
Affinity DataKi:  33nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093118(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  38nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093101(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  39nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093114(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  47nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093113(CHEMBL306097 | N-{1-[2-(4-{5-(3,5-Bis-trifluoromet...)
Affinity DataKi:  48nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093114(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  52nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093117(1-(3,5-Bis-trifluoromethyl-benzyloxy)-5-(4-cyclohe...)
Affinity DataKi:  53nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093108(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  61nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093109(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  62nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093099(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  70nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093122(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093100(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  82nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093111(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  95nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093115(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  113nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093121(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  125nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093119(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  125nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093117(1-(3,5-Bis-trifluoromethyl-benzyloxy)-5-(4-cyclohe...)
Affinity DataKi:  128nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093103(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  136nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093098(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  136nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093122(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093106(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  181nMAssay Description:Inhibitory activity against human tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093108(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  200nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093100(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  208nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093099(1-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4-dichl...)
Affinity DataKi:  217nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093109(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  259nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093102(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  266nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-K receptor(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50093115(2-(4-{5-(3,5-Bis-trifluoromethyl-benzyloxy)-3-(3,4...)
Affinity DataKi:  368nMAssay Description:Inhibitory activity against human tachykinin receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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