Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50010381
TargetAdenosine receptor A2a(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi:  0.0480nMAssay Description:Inhibitory activity against human adenosine A2A receptor expressed in HEK293 cells by displacement of [3H]SCH-58261More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2a(Rat)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi:  0.5nMAssay Description:Inhibitory activity against adenosine A2A receptor in rat striatal membranes by displacement of [3H]SCH-58261More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi:  1.11E+3nMAssay Description:Inhibitory activity against human adenosine A1 receptor expressed in CHO cells by displacement of [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Rat)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi:  1.82E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Rat)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against rat adenosine A3 receptor expressed in HEK293 cells by displacement of [125I]AB-MECAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A2b(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human adenosine A2B receptor expressed in HEK293 cells by displacement of [3H]DPCPXMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed