Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50003567
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473051BDBM50473051(CHEMBL142136)
Affinity DataKi:  0.0500nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50128836BDBM50128836(CHEMBL143228)
Affinity DataKi:  0.0700nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473042BDBM50473042(CHEMBL141269)
Affinity DataKi:  0.160nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473044BDBM50473044(CHEMBL343764)
Affinity DataKi:  0.410nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473039BDBM50473039(CHEMBL423551)
Affinity DataKi:  0.480nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473050BDBM50473050(CHEMBL342839)
Affinity DataKi:  0.660nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473045BDBM50473045(CHEMBL142084)
Affinity DataKi:  0.720nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473047BDBM50473047(CHEMBL139948)
Affinity DataKi:  1.10nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473046BDBM50473046(CHEMBL342669)
Affinity DataKi:  1.5nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473053BDBM50473053(CHEMBL141559)
Affinity DataKi:  1.80nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473067BDBM50473067(CHEMBL343290)
Affinity DataKi:  1.90nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473065BDBM50473065(CHEMBL139610)
Affinity DataKi:  2.30nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473064BDBM50473064(CHEMBL140277)
Affinity DataKi:  2.60nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473066BDBM50473066(CHEMBL141842)
Affinity DataKi:  2.70nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473059BDBM50473059(CHEMBL336052)
Affinity DataKi:  3.90nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473040BDBM50473040(CHEMBL341731)
Affinity DataKi:  4.30nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473056BDBM50473056(CHEMBL141097)
Affinity DataKi:  4.60nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473057BDBM50473057(CHEMBL335339)
Affinity DataKi:  5.20nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473062BDBM50473062(CHEMBL142026)
Affinity DataKi:  6.20nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473043BDBM50473043(CHEMBL140576)
Affinity DataKi:  8.40nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473041BDBM50473041(CHEMBL140993)
Affinity DataKi:  8.70nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473058BDBM50473058(CHEMBL141397)
Affinity DataKi:  9.5nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473055BDBM50473055(CHEMBL343340)
Affinity DataKi:  12nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473048BDBM50473048(CHEMBL421933)
Affinity DataKi:  17nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473063BDBM50473063(CHEMBL141174)
Affinity DataKi:  21nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473049BDBM50473049(CHEMBL141701)
Affinity DataKi:  26nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473038BDBM50473038(CHEMBL337773)
Affinity DataKi:  31nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473054BDBM50473054(CHEMBL140935)
Affinity DataKi:  43nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473060BDBM50473060(CHEMBL140992)
Affinity DataKi:  132nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473061BDBM50473061(CHEMBL141026)
Affinity DataKi:  146nMAssay Description:In vitro for binding affinity for muscarinic acetylcholine receptors in homogenized rat brain in the presence of [3H]scopolamine.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Rat)
University of Michigan Medical School

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473052BDBM50473052(CHEMBL424105)
Affinity DataKi:  237nMAssay Description:Tested in vitro for binding affinity against Muscarinic acetylcholine receptor from rat brain using [3H]- Scopolamine as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed