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Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 50010456
Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095041(CHEMBL328595 | Ethyl-{2-[2-(3-fluoro-phenyl)-1H-in...)
Affinity DataKi:  0.0800nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095043(CHEMBL90911 | Ethyl-methyl-{2-[2-(3-trifluoromethy...)
Affinity DataKi:  0.130nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095035(CHEMBL91549 | Ethyl-methyl-[2-(2-phenyl-1H-indol-3...)
Affinity DataKi:  0.140nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095038(CHEMBL90837 | Ethyl-methyl-{2-[2-(3-nitro-phenyl)-...)
Affinity DataKi:  0.140nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095042(3-[2-((R)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  0.180nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095036(CHEMBL330303 | {2-[2-(3,5-Bis-trifluoromethyl-phen...)
Affinity DataKi:  0.190nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095037(3-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-...)
Affinity DataKi:  0.260nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095044(CHEMBL91197 | Ethyl-{2-[2-(2-fluoro-phenyl)-1H-ind...)
Affinity DataKi:  0.300nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095034(4-{3-[2-(Ethyl-methyl-amino)-ethyl]-1H-indol-2-yl}...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095039(CHEMBL328459 | Ethyl-{2-[2-(4-fluoro-phenyl)-1H-in...)
Affinity DataKi:  0.430nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095033(CHEMBL92416 | Ethyl-methyl-[2-(2-thiophen-2-yl-1H-...)
Affinity DataKi:  1.70nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095028(2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole | CH...)
Affinity DataKi:  2.60nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095034(4-{3-[2-(Ethyl-methyl-amino)-ethyl]-1H-indol-2-yl}...)
Affinity DataKi:  2.60nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095040(CHEMBL328257 | Diethyl-[2-(2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  2.80nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095045(CHEMBL91463 | {2-[2-(4-Chloro-phenyl)-1H-indol-3-y...)
Affinity DataKi:  3.5nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095047(3-[2-((S)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  4nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095029(CHEMBL91447 | Dimethyl-[2-(2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  4.40nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095041(CHEMBL328595 | Ethyl-{2-[2-(3-fluoro-phenyl)-1H-in...)
Affinity DataKi:  8.40nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095031(2-Phenyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole | C...)
Affinity DataKi:  9nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095035(CHEMBL91549 | Ethyl-methyl-[2-(2-phenyl-1H-indol-3...)
Affinity DataKi:  11nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095043(CHEMBL90911 | Ethyl-methyl-{2-[2-(3-trifluoromethy...)
Affinity DataKi:  12nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095036(CHEMBL330303 | {2-[2-(3,5-Bis-trifluoromethyl-phen...)
Affinity DataKi:  15nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095043(CHEMBL90911 | Ethyl-methyl-{2-[2-(3-trifluoromethy...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095039(CHEMBL328459 | Ethyl-{2-[2-(4-fluoro-phenyl)-1H-in...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095042(3-[2-((R)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095037(3-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-...)
Affinity DataKi:  29nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095044(CHEMBL91197 | Ethyl-{2-[2-(2-fluoro-phenyl)-1H-ind...)
Affinity DataKi:  30nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095039(CHEMBL328459 | Ethyl-{2-[2-(4-fluoro-phenyl)-1H-in...)
Affinity DataKi:  31nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095045(CHEMBL91463 | {2-[2-(4-Chloro-phenyl)-1H-indol-3-y...)
Affinity DataKi:  36nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095042(3-[2-((R)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  36nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095038(CHEMBL90837 | Ethyl-methyl-{2-[2-(3-nitro-phenyl)-...)
Affinity DataKi:  36nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095038(CHEMBL90837 | Ethyl-methyl-{2-[2-(3-nitro-phenyl)-...)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095032(3-(2-Azetidin-1-yl-ethyl)-2-phenyl-1H-indole | CHE...)
Affinity DataKi:  44nMAssay Description:Displacent of [H]-ketanserin from CHO cells expressing human 5-hydroxytryptamine 2A receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095041(CHEMBL328595 | Ethyl-{2-[2-(3-fluoro-phenyl)-1H-in...)
Affinity DataKi:  68nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095033(CHEMBL92416 | Ethyl-methyl-[2-(2-thiophen-2-yl-1H-...)
Affinity DataKi:  78nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095035(CHEMBL91549 | Ethyl-methyl-[2-(2-phenyl-1H-indol-3...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095037(3-[2-((S)-2-Methoxymethyl-pyrrolidin-1-yl)-ethyl]-...)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095033(CHEMBL92416 | Ethyl-methyl-[2-(2-thiophen-2-yl-1H-...)
Affinity DataKi:  120nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095044(CHEMBL91197 | Ethyl-{2-[2-(2-fluoro-phenyl)-1H-ind...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095034(4-{3-[2-(Ethyl-methyl-amino)-ethyl]-1H-indol-2-yl}...)
Affinity DataKi:  160nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095040(CHEMBL328257 | Diethyl-[2-(2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  160nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095029(CHEMBL91447 | Dimethyl-[2-(2-phenyl-1H-indol-3-yl)...)
Affinity DataKi:  180nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095036(CHEMBL330303 | {2-[2-(3,5-Bis-trifluoromethyl-phen...)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095047(3-[2-((S)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  230nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095045(CHEMBL91463 | {2-[2-(4-Chloro-phenyl)-1H-indol-3-y...)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095031(2-Phenyl-3-(2-pyrrolidin-1-yl-ethyl)-1H-indole | C...)
Affinity DataKi:  260nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2C(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095028(2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole | CH...)
Affinity DataKi:  268nMAssay Description:Displacement of [H]-mesulergine from CHO cells expressing human 5-hydroxytryptamine 2C receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095047(3-[2-((S)-2-Methyl-piperidin-1-yl)-ethyl]-2-phenyl...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095028(2-Phenyl-3-(2-piperidin-1-yl-ethyl)-1H-indole | CH...)
Affinity DataKi:  896nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Human)
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50095032(3-(2-Azetidin-1-yl-ethyl)-2-phenyl-1H-indole | CHE...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-spiperone from CHO cells expressing human Dopamine receptor D2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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