TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 0.745nMAssay Description:Displacement of [3H]-N6-PIA binding from A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 486nMAssay Description:Displacement of [3H]-N6-PIA (Kd, 1 nM) binding from Adenosine A1 receptor in whole rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 648nMAssay Description:Displacement of [3H]-CGS-21,680 (Kd, 14.9 nM) from A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 930nMAssay Description:Displacement of [3H]-CGS-21,680 (Kd, 14.9 nM) from A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Astrazeneca R&D Griffith University
Curated by ChEMBL
Astrazeneca R&D Griffith University
Curated by ChEMBL
Affinity DataKi: 2.12E+3nMAssay Description:Displacement of [3H]-CGS-21,680 (Kd, 14.9 nM) from A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair