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Found 6 Enz. Inhib. hit(s) with all data for entry = 50010592
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  15nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7...)
Affinity DataKi:  46nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7...)
Affinity DataKi:  91nMAssay Description:Binding affinity for protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7...)
Affinity DataKi:  121nMAssay Description:Binding affinity for protein kinase C epsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  334nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096602((2S,5S)-5-Hydroxymethyl-2-isopropyl-7-methoxy-1-me...)
Affinity DataKi:  7.16E+3nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed