Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50010636
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096914BDBM50096914(8-Methyl-3-(1-methyl-1H-indol-5-yl)-8-aza-bicyclo[...)
Affinity DataIC50: 0.75nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096921BDBM50096921(3-[4-(1-Methyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096913BDBM50096913(3-(1-Ethyl-1H-indol-5-yl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096922BDBM50096922(3-(1-Methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096915BDBM50096915(3-(1-Ethyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octa...)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096922BDBM50096922(3-(1-Methyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]oct...)
Affinity DataIC50: 2.70nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096914BDBM50096914(8-Methyl-3-(1-methyl-1H-indol-5-yl)-8-aza-bicyclo[...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096915BDBM50096915(3-(1-Ethyl-1H-indol-5-yl)-8-aza-bicyclo[3.2.1]octa...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096913BDBM50096913(3-(1-Ethyl-1H-indol-5-yl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096916BDBM50096916(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096926BDBM50096926(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicycl...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096919BDBM50096919(8-Methyl-3-[4-(1-methyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096916BDBM50096916(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096918BDBM50096918(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096923BDBM50096923(3-[4-(1,5-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096920BDBM50096920(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-...)
Affinity DataIC50: 58nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096920BDBM50096920(3-[4-(1-Benzyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-...)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096925BDBM50096925(3-[4-(1-Methyl-5-phenyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096924BDBM50096924(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-a...)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096921BDBM50096921(3-[4-(1-Methyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicyc...)
Affinity DataIC50: 614nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096919BDBM50096919(8-Methyl-3-[4-(1-methyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataIC50: 703nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096923BDBM50096923(3-[4-(1,5-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataIC50: 825nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096917BDBM50096917(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-methy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096926BDBM50096926(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-bicycl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096925BDBM50096925(3-[4-(1-Methyl-5-phenyl-1H-pyrrol-2-yl)-phenyl]-8-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096917BDBM50096917(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-methy...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]paroxetine from Serotonin transporter of rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096924BDBM50096924(3-[4-(1-Ethyl-1H-pyrrol-2-yl)-phenyl]-8-methyl-8-a...)
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
State University of New York

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50096918BDBM50096918(3-[4-(1,3-Dimethyl-1H-pyrrol-2-yl)-phenyl]-8-aza-b...)
Affinity DataIC50: 1.47E+3nMAssay Description:Displacement of [125I]RTI-55 from Dopamine transporter of rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed