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Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50041305
TargetBeta-2 adrenergic receptor(Dog)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataIC50:  0.100nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. IC50, the mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002133((+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydrox...)
Affinity DataIC50:  9.12nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM97162(MLS002153782 | RITODRINE | RITODRINE HYDROCHLORIDE...)
Affinity DataIC50:  24.0nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409479(CHEMBL32933)
Affinity DataIC50:  61.7nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409484(CHEMBL32470)
Affinity DataIC50:  251nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409476(CHEMBL289670)
Affinity DataIC50:  282nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409470(CHEMBL32532)
Affinity DataIC50:  646nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409469(CHEMBL284520)
Affinity DataIC50:  1.29E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409471(CHEMBL32586)
Affinity DataIC50:  1.41E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409475(CHEMBL32939)
Affinity DataIC50:  1.41E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409480(CHEMBL33360)
Affinity DataIC50:  1.58E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409478(CHEMBL285888)
Affinity DataIC50:  1.70E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409481(CHEMBL35738)
Affinity DataIC50:  2.19E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409473(CHEMBL33399)
Affinity DataIC50:  2.57E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409468(CHEMBL32670)
Affinity DataIC50:  3.31E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002134(5-((2R)-2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl...)
Affinity DataIC50:  9.77E+3nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409482(CHEMBL35459)
Affinity DataIC50:  1.10E+4nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-2 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409472(CHEMBL32391)
Affinity DataIC50:  1.41E+4nMAssay Description:Agonistic activity towards beta-2 adrenoceptor. Mean concentration required to produce 50% inhibition of uterine contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409479(CHEMBL32933)
Affinity DataEC50:  7.24nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409470(CHEMBL32532)
Affinity DataEC50:  24.0nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409482(CHEMBL35459)
Affinity DataEC50:  22.9nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409481(CHEMBL35738)
Affinity DataEC50:  813nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409484(CHEMBL32470)
Affinity DataEC50:  12.9nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409483(CHEMBL32115)
Affinity DataEC50:  11.0nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409480(CHEMBL33360)
Affinity DataEC50:  52.5nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409476(CHEMBL289670)
Affinity DataEC50:  832nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002134(5-((2R)-2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl...)
Affinity DataEC50:  25.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409478(CHEMBL285888)
Affinity DataEC50:  457nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409468(CHEMBL32670)
Affinity DataEC50:  0.933nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM97162(MLS002153782 | RITODRINE | RITODRINE HYDROCHLORIDE...)
Affinity DataEC50:  191nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50002133((+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydrox...)
Affinity DataEC50:  2.19nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataEC50:  87.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. EC50, the mean concentration required to produce 50% relaxation of detrusor before the addition in th...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409475(CHEMBL32939)
Affinity DataEC50:  575nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409474(CHEMBL417137)
Affinity DataEC50:  158nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409473(CHEMBL33399)
Affinity DataEC50:  81.3nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409472(CHEMBL32391)
Affinity DataEC50:  14.1nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409471(CHEMBL32586)
Affinity DataEC50:  5.62nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetBeta-3 adrenergic receptor(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50409469(CHEMBL284520)
Affinity DataEC50:  61.7nMAssay Description:Agonistic activity towards beta-3 adrenoceptor. Mean concentration required to produce 50% relaxation of detrusor before the addition in the ferret d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed