Compile Data Set for Download or QSAR
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Found 16 Enz. Inhib. hit(s) with all data for entry = 50010815
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  27nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099028(1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50:  28nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099017(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  36nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099025(CHEMBL11011 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099022(CHEMBL268479 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)...)
Affinity DataIC50:  47nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099024(1-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50:  48nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of human Gonadotropin-releasing hormone receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099021(CHEMBL11370 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099029(CHEMBL10941 | Ethanesulfonic acid [4-(4-{2-[2-(3,5...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099020(CHEMBL11156 | Propane-2-sulfonic acid [4-(4-{2-[2-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099027(CHEMBL11074 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099019(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099026(CHEMBL11067 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  300nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  357nMAssay Description:Inhibition of human Gonadotropin-releasing hormone receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099018(CHEMBL273296 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  500nMAssay Description:Inhibition of rat GnRH receptor bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed