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Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50010816
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  7nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099036(CHEMBL11009 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  16nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  27nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099041(CHEMBL11014 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  36nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099033(CHEMBL262715 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  40nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099051(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  41nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099045(CHEMBL273625 | N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)...)
Affinity DataIC50:  45nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099043(CHEMBL11253 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099046(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  57nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099040(CHEMBL11310 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  90nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099030(CHEMBL11263 | N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099050(CHEMBL11420 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  150nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099042(CHEMBL275287 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  160nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099023(CHEMBL11149 | N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-...)
Affinity DataIC50:  170nMAssay Description:Inhibitory activity of the compound evaluated against human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099034(CHEMBL11021 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099048(CHEMBL11436 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  200nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099032(CHEMBL273725 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  210nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099037(CHEMBL275920 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  270nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50:  357nMAssay Description:Inhibitory activity of the compound evaluated against human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099044(CHEMBL11375 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099039(CHEMBL11087 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  450nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099038(CHEMBL11623 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099035(CHEMBL269636 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50:  2.17E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099047(CHEMBL11523 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099049(CHEMBL11134 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indol...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50099031(CHEMBL274441 | {2-[2-(3,5-Dimethyl-phenyl)-1H-indo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed