Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50010816
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099023BDBM50099023(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 7nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099036BDBM50099036({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 16nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097007BDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 27nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099041BDBM50099041({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 36nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099033BDBM50099033({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 40nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099051BDBM50099051(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 41nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099045BDBM50099045(N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 45nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099043BDBM50099043({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 50nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099046BDBM50099046(5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 57nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099040BDBM50099040({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099030BDBM50099030(N-[5-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 120nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099050BDBM50099050({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 150nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099042BDBM50099042({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 160nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099023BDBM50099023(N-[4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity evaluated against human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099034BDBM50099034({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099048BDBM50099048({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099032BDBM50099032({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099037BDBM50099037({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 270nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50097007BDBM50097007(4-(4-{2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-et...)
Affinity DataIC50: 357nMAssay Description:Inhibitory activity evaluated against human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099044BDBM50099044({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 450nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099039BDBM50099039({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 450nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099038BDBM50099038({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099035BDBM50099035({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099047BDBM50099047({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099049BDBM50099049({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50099031BDBM50099031({2-[2-(3,5-Dimethyl-phenyl)-1H-indol-3-yl]-ethyl}-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed