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Report error Found 254 Enz. Inhib. hit(s) with all data for entry = 50010899
TargetD(4) dopamine receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  0.430nMAssay Description:In vitro binding affinity to human Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099893(3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  2.30nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099889(3-[4-(4-Vinyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  2.80nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099887(3-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  3.30nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50075360(3-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  3.60nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  3.70nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099892(3-[4-(4-Methylsulfanyl-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  4.70nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  5nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099894(3-[4-(4-Propyl-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  6.70nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099891(3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  34nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099892(3-[4-(4-Methylsulfanyl-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity to cloned rat Dopamine receptor D3 measured by displacement of the radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  103nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(4) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099895(3-(4-Biphenyl-4-yl-piperazin-1-ylmethyl)-1H-pyrrol...)
Affinity DataKi:  148nMAssay Description:In vitro binding affinity to rat Dopamine receptor D4 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099887(3-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  213nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  226nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099893(3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  232nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099887(3-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  242nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099891(3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  318nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099892(3-[4-(4-Methylsulfanyl-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi:  336nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  406nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  411nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099893(3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  412nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(2) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  438nMAssay Description:In vitro binding affinity to rat Dopamine receptor D2 measured by displacement of the radioligand [3H]-spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  453nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099889(3-[4-(4-Vinyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  509nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  627nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  668nMAssay Description:In vitro binding affinity to cloned rat Dopamine receptor D3 measured by displacement of the radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 7(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099894(3-[4-(4-Propyl-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  713nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 7 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099894(3-[4-(4-Propyl-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  921nMAssay Description:In vitro binding affinity to cloned rat Dopamine receptor D3 measured by displacement of the radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099887(3-[4-(2-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  991nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  1.66E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetD(3) dopamine receptor(Rat)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  1.69E+3nMAssay Description:In vitro binding affinity to cloned rat Dopamine receptor D3 measured by displacement of the radioligand [3H]-sulpirideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099895(3-(4-Biphenyl-4-yl-piperazin-1-ylmethyl)-1H-pyrrol...)
Affinity DataKi:  1.93E+3nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  2.31E+3nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099893(3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  2.76E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 2A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099891(3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  2.79E+3nMAssay Description:Binding affinity to cloned human 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099889(3-[4-(4-Vinyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  3.97E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi:  4.46E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099894(3-[4-(4-Propyl-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi:  6.49E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 1A(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM85093(CAS_3853 | CHEMBL267014 | CHEMBL555670 | L 745,870...)
Affinity DataKi:  6.62E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099891(3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi:  7.11E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 6(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi:  7.39E+3nMAssay Description:In vitro binding affinity to human 5-hydroxytryptamine 6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50075360(3-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099891(3-[4-(4-Trifluoromethyl-phenyl)-piperazin-1-ylmeth...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099889(3-[4-(4-Vinyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099890(3-[4-(2-Methoxy-phenyl)-piperazin-1-ylmethyl]-1H-p...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099893(3-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-1H-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099888(3-[4-(4-Ethyl-phenyl)-piperazin-1-ylmethyl]-1H-pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
Columbia University College of Physicians and Surgeons

Curated by ChEMBL
LigandPNGBDBM50099892(3-[4-(4-Methylsulfanyl-phenyl)-piperazin-1-ylmethy...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to cloned Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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