Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50011308
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105035BDBM50105035(N-{5-Benzo[1,3]dioxol-5-yl-6-[2-(5-methylsulfanyl-...)
Affinity DataIC50: 0.00110nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105034BDBM50105034(4-tert-Butyl-N-{6-[2-(5-methoxy-pyrimidin-2-yloxy)...)
Affinity DataIC50: 0.00170nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104997BDBM50104997(4-tert-Butyl-N-[6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50: 0.00170nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105048BDBM50105048(N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-(2-m...)
Affinity DataIC50: 0.00390nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105047BDBM50105047(Acetic acid ethyl ester4-tert-Butyl-N-{5-(3,4-dime...)
Affinity DataIC50: 0.00850nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104986BDBM50104986(4-tert-Butyl-N-{5-(4-ethyl-phenyl)-6-[2-(5-methyls...)
Affinity DataIC50: 0.0130nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105040BDBM50105040(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(5-meth...)
Affinity DataIC50: 0.0150nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105026BDBM50105026(N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-(2-m...)
Affinity DataIC50: 0.0180nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105025BDBM50105025(4-tert-Butyl-N-{5-(3-methoxy-phenyl)-6-[2-(5-methy...)
Affinity DataIC50: 0.0280nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104988BDBM50104988(4-tert-Butyl-N-{6-[2-(5-pyridin-2-yl-pyrimidin-2-y...)
Affinity DataIC50: 0.0360nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104995BDBM50104995(sodium salt of N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)...)
Affinity DataIC50: 0.0390nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104992BDBM50104992(N-[6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-(3-m...)
Affinity DataIC50: 0.0510nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104991BDBM50104991(4-tert-Butyl-N-[6-[2-(5-chloro-pyrimidin-2-yloxy)-...)
Affinity DataIC50: 0.0590nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105027BDBM50105027(sodium salt of 4-tert-Butyl-N-{6-[2-(5-chloro-pyri...)
Affinity DataIC50: 0.0800nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105042BDBM50105042(4-tert-Butyl-N-{6-[2-(pyrimidin-2-yloxy)-ethoxy]-5...)
Affinity DataIC50: 0.110nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105029BDBM50105029(4-tert-Butyl-N-[6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105007BDBM50105007(N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-to...)
Affinity DataIC50: 0.160nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104987BDBM50104987(sodium salt of 4-tert-Butyl-N-{6-[2-(5-thiophen-2-...)
Affinity DataIC50: 0.25nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104984BDBM50104984(4-tert-Butyl-N-{6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50: 0.290nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105003BDBM50105003(4-tert-Butyl-N-{5-(2-methoxy-phenoxy)-6-[2-(5-meth...)
Affinity DataIC50: 0.370nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104993BDBM50104993(sodium salt of 4-tert-Butyl-N-{6-[2-(5-methylsulfa...)
Affinity DataIC50: 0.420nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104982BDBM50104982(sodium salt of 4-tert-Butyl-N-{6-[2-(5-furan-2-yl-...)
Affinity DataIC50: 0.480nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105011BDBM50105011(sodium salt of 4-tert-Butyl-N-{6-[2-(5-methoxy-pyr...)
Affinity DataIC50: 0.560nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105041BDBM50105041(N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-to...)
Affinity DataIC50: 0.640nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105019BDBM50105019(N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-to...)
Affinity DataIC50: 0.760nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105002BDBM50105002(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(5-meth...)
Affinity DataIC50: 0.860nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104983BDBM50104983(4-tert-Butyl-N-{6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50: 0.890nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105046BDBM50105046(Naphthalene-2-sulfonic acid {6-[2-(5-bromo-pyrimid...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105014BDBM50105014(N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-to...)
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105038BDBM50105038(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyrimi...)
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105021BDBM50105021(4-tert-Butyl-N-{5-(4-isopropyl-phenyl)-6-[2-(5-met...)
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Rat)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105000BDBM50105000(sodium salt of 4-tert-Butyl-N-[6-(2-hydroxy-ethoxy...)
Affinity DataIC50: 1.40nMAssay Description:In vitro for specific binding of [125I]ET1 to A10 cell expressed in endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105032BDBM50105032(N-{6-[2-(5-Bromo-pyrimidin-2-yloxy)-ethoxy]-5-p-to...)
Affinity DataIC50: 1.40nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104990BDBM50104990(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyrimi...)
Affinity DataIC50: 1.90nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105043BDBM50105043(1,2,3,4-Tetrahydro-fluoren-9-one salt ofN-{6-[2-(5...)
Affinity DataIC50: 1.90nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104996BDBM50104996(4-Bromo-N-{6-[2-(5-bromo-pyrimidin-2-yloxy)-ethoxy...)
Affinity DataIC50: 2.80nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104994BDBM50104994(4-tert-Butyl-N-{5-furan-2-yl-6-[2-(5-methylsulfany...)
Affinity DataIC50: 2.90nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104999BDBM50104999(Thiophene-2-sulfonic acid {6-[2-(5-bromo-pyrimidin...)
Affinity DataIC50: 3.10nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105020BDBM50105020(5-Pyridin-2-yl-thiophene-2-sulfonic acid {6-[2-(5-...)
Affinity DataIC50: 3.40nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104987BDBM50104987(sodium salt of 4-tert-Butyl-N-{6-[2-(5-thiophen-2-...)
Affinity DataIC50: 3.80nMAssay Description:In vitro for specific binding of [125I]ET1 to GHcell expressed in Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105045BDBM50105045(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyrimi...)
Affinity DataIC50: 6.20nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin receptor type B(Human)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50104982BDBM50104982(sodium salt of 4-tert-Butyl-N-{6-[2-(5-furan-2-yl-...)
Affinity DataIC50: 7nMAssay Description:In vitro for specific binding of [125I]ET1 to GHcell expressed in Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105000BDBM50105000(sodium salt of 4-tert-Butyl-N-[6-(2-hydroxy-ethoxy...)
Affinity DataIC50: 7.5nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105037BDBM50105037(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyridi...)
Affinity DataIC50: 8.80nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105016BDBM50105016(4-tert-Butyl-N-{6-[2-(5-methylsulfanyl-pyrimidin-2...)
Affinity DataIC50: 9.90nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105001BDBM50105001(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(thiazo...)
Affinity DataIC50: 12nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105012BDBM50105012(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(quinol...)
Affinity DataIC50: 15.2nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105030BDBM50105030(Naphthalene-1-sulfonic acid {6-[2-(5-bromo-pyrimid...)
Affinity DataIC50: 22nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105018BDBM50105018(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyrazi...)
Affinity DataIC50: 24.5nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Tanabe Seiyaku

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50105044BDBM50105044(4-tert-Butyl-N-{5-(3-methoxy-phenoxy)-6-[2-(pyrimi...)
Affinity DataIC50: 25.8nMAssay Description:In vitro inhibition of [125I]ET1 binding to Endothelin A receptor in porcine aortic membrane from endothelial cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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