Compile Data Set for Download or QSAR
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Report error Found 44 Enz. Inhib. hit(s) with all data for entry = 50011447
TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106632(4-[2-(4-hydroxyphenyl)-3-butynyl]phenol | CHEMBL33...)
Affinity DataEC50:  3.10nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.0180nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106634((S)-3-(4-Hydroxy-phenyl)-2-((R)-4-hydroxy-phenyl)-...)
Affinity DataEC50:  0.140nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106635((+/-)-2,3-bis(4-hydroxyphenyl)propanenitrile | 2,3...)
Affinity DataEC50:  20nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106636(2,3-Bis-(4-hydroxy-phenyl)-propionic acid methyl e...)
Affinity DataEC50:  2.70nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106637(4-[2-(4-hydroxyphenyl)-3-pentynyl]phenol | CHEMBL1...)
Affinity DataEC50:  2.10nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106638(2,3-Bis-(4-hydroxy-phenyl)-2-methyl-propionitrile ...)
Affinity DataEC50:  8nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106638(2,3-Bis-(4-hydroxy-phenyl)-2-methyl-propionitrile ...)
Affinity DataEC50:  23nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106639(1,1,1-Trifluoro-3,4-bis-(4-hydroxy-phenyl)-butan-2...)
Affinity DataEC50:  160nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  6nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106640(4-[3,3,4,4,4-pentafluoro-2-(4-hydroxyphenyl)butyl]...)
Affinity DataEC50:  15nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106642(4-[3,3,3-trifluoro-2-(4-hydroxyphenyl)propyl]pheno...)
Affinity DataEC50:  2nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106641(2,3-Bis-(4-hydroxy-phenyl)-acrylonitrile | CHEMBL3...)
Affinity DataEC50:  95nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106634((S)-3-(4-Hydroxy-phenyl)-2-((R)-4-hydroxy-phenyl)-...)
Affinity DataEC50:  5.20nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM19459(5,7-dihydroxy-3-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataEC50:  20nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106643(3-(4-Hydroxy-2-methyl-phenyl)-2-(4-hydroxy-phenyl)...)
Affinity DataEC50:  0.370nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106644(2,3-Bis-(4-hydroxy-phenyl)-succinonitrile | CHEMBL...)
Affinity DataEC50:  14nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106646((S)-3-(4-Hydroxy-phenyl)-2-((R)-4-hydroxy-phenyl)-...)
Affinity DataEC50:  0.0640nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106641(2,3-Bis-(4-hydroxy-phenyl)-acrylonitrile | CHEMBL3...)
Affinity DataEC50:  140nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106646((S)-3-(4-Hydroxy-phenyl)-2-((R)-4-hydroxy-phenyl)-...)
Affinity DataEC50:  0.150nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106632(4-[2-(4-hydroxyphenyl)-3-butynyl]phenol | CHEMBL33...)
Affinity DataEC50:  1.40nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106645(2-(4-Hydroxy-2-methyl-phenyl)-3-(4-hydroxy-phenyl)...)
Affinity DataEC50:  1.70nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106640(4-[3,3,4,4,4-pentafluoro-2-(4-hydroxyphenyl)butyl]...)
Affinity DataEC50:  42nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106642(4-[3,3,3-trifluoro-2-(4-hydroxyphenyl)propyl]pheno...)
Affinity DataEC50:  2.90nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106633(3,4-Bis-(4-hydroxy-phenyl)-butyronitrile | CHEMBL1...)
Affinity DataEC50:  30nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106645(2-(4-Hydroxy-2-methyl-phenyl)-3-(4-hydroxy-phenyl)...)
Affinity DataEC50:  16nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106636(2,3-Bis-(4-hydroxy-phenyl)-propionic acid methyl e...)
Affinity DataEC50:  4.90nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106647(2-(4-Hydroxy-phenyl)-3-(3-hydroxy-phenyl)-succinon...)
Affinity DataEC50:  110nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106644(2,3-Bis-(4-hydroxy-phenyl)-succinonitrile | CHEMBL...)
Affinity DataEC50:  0.420nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106643(3-(4-Hydroxy-2-methyl-phenyl)-2-(4-hydroxy-phenyl)...)
Affinity DataEC50:  6.70nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106648(2-(4-Hydroxy-benzyl)-2-(4-hydroxy-phenyl)-malononi...)
Affinity DataEC50:  21nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106635((+/-)-2,3-bis(4-hydroxyphenyl)propanenitrile | 2,3...)
Affinity DataEC50:  6nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106644(2,3-Bis-(4-hydroxy-phenyl)-succinonitrile | CHEMBL...)
Affinity DataEC50:  14nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106647(2-(4-Hydroxy-phenyl)-3-(3-hydroxy-phenyl)-succinon...)
Affinity DataEC50:  150nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106639(1,1,1-Trifluoro-3,4-bis-(4-hydroxy-phenyl)-butan-2...)
Affinity DataEC50:  464nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106644(2,3-Bis-(4-hydroxy-phenyl)-succinonitrile | CHEMBL...)
Affinity DataEC50:  0.410nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106648(2-(4-Hydroxy-benzyl)-2-(4-hydroxy-phenyl)-malononi...)
Affinity DataEC50:  40nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106650(3,4-Bis-(4-hydroxy-phenyl)-butan-2-one | CHEMBL135...)
Affinity DataEC50:  18nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106649(4-[1-(1-ethynyl)-2-(4-hydroxyphenyl)-3-butynyl]phe...)
Affinity DataEC50:  73nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106649(4-[1-(1-ethynyl)-2-(4-hydroxyphenyl)-3-butynyl]phe...)
Affinity DataEC50:  3.70nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106650(3,4-Bis-(4-hydroxy-phenyl)-butan-2-one | CHEMBL135...)
Affinity DataEC50:  35nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106637(4-[2-(4-hydroxyphenyl)-3-pentynyl]phenol | CHEMBL1...)
Affinity DataEC50:  0.380nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEstrogen receptor beta(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataEC50:  0.0390nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor BetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetEstrogen receptor(Human)
University of Illinois

Curated by ChEMBL
LigandPNGBDBM50106633(3,4-Bis-(4-hydroxy-phenyl)-butyronitrile | CHEMBL1...)
Affinity DataEC50:  130nMAssay Description:Transcriptional potency (EC50) at Human estrogen receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed