Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50011686
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109332(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50: 120nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109338(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50: 150nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109319(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propyl-py...)
Affinity DataIC50: 220nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109316(1-[4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyr...)
Affinity DataIC50: 240nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109337(1-[5-Butyl-4-(4-fluoro-phenyl)-2,6-diisopropyl-pyr...)
Affinity DataIC50: 250nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109339(1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-py...)
Affinity DataIC50: 300nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109329([4-(4-Fluoro-phenyl)-5-hexyl-2,6-diisopropyl-pyrid...)
Affinity DataIC50: 350nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109323([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propyl-pyri...)
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109341([4-(4-Fluoro-phenyl)-5-heptyl-2,6-diisopropyl-pyri...)
Affinity DataIC50: 700nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-pentyl-pyri...)
Affinity DataIC50: 700nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109318([5-Butyl-4-(4-fluoro-phenyl)-2,6-diisopropyl-pyrid...)
Affinity DataIC50: 750nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109325([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(3-methyl-b...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109327([5-Ethyl-4-(4-fluoro-phenyl)-2,6-diisopropyl-pyrid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109315([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-octyl-pyrid...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109317((5-Ethyl-2,6-diisopropyl-4-phenyl-pyridin-3-yl)-me...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-p...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109330([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-vinyl-pyrid...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109322([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-p...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibitory concentration against binding to the human glucagon receptor (hGR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109321([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-methyl-pyri...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109320([4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-methoxymeth...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109324(4-(4-Fluoro-phenyl)-5-hydroxymethyl-2,6-diisopropy...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109328((2,6-Dimethyl-5-pentyl-4-phenyl-pyridin-3-yl)-meth...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109333([4-(4-Fluoro-phenyl)-5-hydroxymethyl-2,6-diisoprop...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109334((2,6-Diethyl-5-pentyl-4-phenyl-pyridin-3-yl)-metha...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109335((2,5,6-Triethyl-4-phenyl-pyridin-3-yl)-methanol | ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlucagon receptor(Human)
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109340((5-Ethyl-2,6-dimethyl-4-phenyl-pyridin-3-yl)-metha...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration against cAMP production in hGR-CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed