Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50011738
LigandPNGBDBM50109937((R)-2-[(Indane-2-carbonyl)-amino]-3-naphthalen-1-y...)
Affinity DataIC50:  7.30nMAssay Description:Tested for the inhibition of Candida GGTase I in Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109938(9H-Xanthene-9-carboxylic acid {(R)-2-(3,4-dichloro...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Candida geranylgeranyl transferase I at 3 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109933(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  17nMAssay Description:Tested for the inhibition of Candida GGTase I in Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109933(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  17nMAssay Description:Tested for the inhibition of Candida GGTase I in Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109940(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  31nMAssay Description:Tested for the inhibition of Candida GGTase I in Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109935(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  240nMAssay Description:Inhibition of Candida geranylgeranyl transferase I at 3 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109934(CHEMBL347650 | Indan-2-carboxylic acid {(R)-1-[2-(...)
Affinity DataIC50:  350nMAssay Description:Inhibition of Candida geranylgeranyl transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109936(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  780nMAssay Description:Tested for the inhibition of Candida GGTase I in Candida albicansMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109939(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of Candida geranylgeranyl transferase I at 3 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109933(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of human geranylgeranyl transferase IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Banyu Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50109933(2-(2,3-Dihydro-benzo[1,4]dioxin-2-yl)-thiazole-4-c...)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed