Compile Data Set for Download or QSAR
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Found 19 Enz. Inhib. hit(s) with all data for entry = 50011953
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  65nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109326((R)-1-[4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-propy...)
Affinity DataIC50:  110nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  120nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112476(5-Fluoro-2-(3-hydroxymethyl-2,6-diisopropyl-5-pent...)
Affinity DataIC50:  190nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  400nMAssay Description:Tested for its ability to inhibit cAMP production in human glucagon receptor expressed CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112484(2-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridi...)
Affinity DataIC50:  500nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109331(CHEMBL24616 | [4-(4-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  700nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112475(CHEMBL286098 | [4-(4-Chloro-phenyl)-2,6-diisopropy...)
Affinity DataIC50:  800nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112479((2,6-Diisopropyl-5-pentyl-4-p-tolyl-pyridin-3-yl)-...)
Affinity DataIC50:  1.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112478(CHEMBL286555 | [4-(3,4-Difluoro-phenyl)-2,6-diisop...)
Affinity DataIC50:  1.10E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50109336((2,6-Diisopropyl-5-pentyl-4-phenyl-pyridin-3-yl)-m...)
Affinity DataIC50:  1.40E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112485(CHEMBL277627 | [4-(2-Amino-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  2.30E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112483(CHEMBL25137 | [4-(3-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  3.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112481(3-(3-Hydroxymethyl-2,6-diisopropyl-5-pentyl-pyridi...)
Affinity DataIC50:  6.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112477(4-(4-Fluoro-phenyl)-2,6-diisopropyl-5-(2-methyl-pr...)
Affinity DataIC50:  7.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112480(CHEMBL25255 | [4-(2-Fluoro-phenyl)-2,6-diisopropyl...)
Affinity DataIC50:  9.00E+3nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112482(CHEMBL24905 | [4-(2,4-Difluoro-phenyl)-2,6-diisopr...)
Affinity DataIC50:  1.10E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112473(CHEMBL24527 | [4-(4-Fluoro-3-hydroxymethyl-phenyl)...)
Affinity DataIC50:  1.90E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Bayer Research Center

Curated by ChEMBL
LigandPNGBDBM50112474(CHEMBL284699 | [2,6-Diisopropyl-4-(3-methoxy-pheny...)
Affinity DataIC50:  4.80E+4nMAssay Description:Tested for its inhibitory activity against human glucagon receptor (hGR) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed