Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 50003603
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21392BDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataKi:  0.490nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403759BDBM50403759(CHEMBL428494)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50116963BDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473640BDBM50473640(CHEMBL71847)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403770BDBM50403770(CHEMBL12427)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50220558BDBM50220558(CHEMBL418888)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50130276BDBM50130276(N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tetrahydro-3H-benz...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403768BDBM50403768(CHEMBL273246)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403780BDBM50403780(CHEMBL12846)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473633BDBM50473633(CHEMBL304731)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403777BDBM50403777(CHEMBL12702)
Affinity DataKi:  5.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473658BDBM50473658(CHEMBL71383)
Affinity DataKi:  5.80nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473644BDBM50473644(CHEMBL302766)
Affinity DataKi:  6nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473648BDBM50473648(CHEMBL71225)
Affinity DataKi:  6.5nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473651BDBM50473651(CHEMBL71959)
Affinity DataKi:  7.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473639BDBM50473639(CHEMBL303166)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473652BDBM50473652(CHEMBL422587)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473657BDBM50473657(CHEMBL70889)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473650BDBM50473650(CHEMBL304167)
Affinity DataKi:  10nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473653BDBM50473653(CHEMBL71057)
Affinity DataKi:  12nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473641BDBM50473641(CHEMBL307101)
Affinity DataKi:  12nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473637BDBM50473637(CHEMBL68094)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473636BDBM50473636(CHEMBL70869)
Affinity DataKi:  17nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473649BDBM50473649(CHEMBL71224)
Affinity DataKi:  17nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473638BDBM50473638(CHEMBL305526)
Affinity DataKi:  19nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473634BDBM50473634(CHEMBL71170)
Affinity DataKi:  19nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473660BDBM50473660(CHEMBL71390)
Affinity DataKi:  20nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473654BDBM50473654(CHEMBL307352)
Affinity DataKi:  22nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473643BDBM50473643(CHEMBL69040)
Affinity DataKi:  24nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473635BDBM50473635(CHEMBL70819)
Affinity DataKi:  25nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473642BDBM50473642(CHEMBL70048)
Affinity DataKi:  28nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473662BDBM50473662(CHEMBL308461)
Affinity DataKi:  30nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473652BDBM50473652(CHEMBL422587)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403770BDBM50403770(CHEMBL12427)
Affinity DataKi:  43nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473646BDBM50473646(CHEMBL302093)
Affinity DataKi:  44nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473650BDBM50473650(CHEMBL304167)
Affinity DataKi:  45nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473656BDBM50473656(CHEMBL72008)
Affinity DataKi:  46nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473643BDBM50473643(CHEMBL69040)
Affinity DataKi:  46nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403759BDBM50403759(CHEMBL428494)
Affinity DataKi:  54nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473640BDBM50473640(CHEMBL71847)
Affinity DataKi:  65nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473645BDBM50473645(CHEMBL307686)
Affinity DataKi:  72nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473655BDBM50473655(CHEMBL69388)
Affinity DataKi:  74nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473647BDBM50473647(CHEMBL71165)
Affinity DataKi:  76nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50220558BDBM50220558(CHEMBL418888)
Affinity DataKi:  79nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473641BDBM50473641(CHEMBL307101)
Affinity DataKi:  98nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473645BDBM50473645(CHEMBL307686)
Affinity DataKi:  98nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50116963BDBM50116963(2a-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-butyl...)
Affinity DataKi:  98nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473647BDBM50473647(CHEMBL71165)
Affinity DataKi:  98nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50403768BDBM50403768(CHEMBL273246)
Affinity DataKi:  105nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Meiji Seika Kaisha

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50473642BDBM50473642(CHEMBL70048)
Affinity DataKi:  110nMAssay Description:Binding affinity to human recombinant 5-hydroxytryptamine 7 receptor in mammalian cells using [3H]5-CT as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
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