Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50012029
TargetC-X-C chemokine receptor type 2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102222BDBM50102222(1-(2-Bromo-phenyl)-3-(7-cyano-3H-benzotriazol-4-yl...)
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113628BDBM50113628([5-(4-Fluoro-phenylcarbamoyl)-pyridin-2-ylsulfanyl...)
Affinity DataIC50: 32nMAssay Description:Displacement of [125I]IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113628BDBM50113628([5-(4-Fluoro-phenylcarbamoyl)-pyridin-2-ylsulfanyl...)
Affinity DataIC50: 42nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219799BDBM50219799(CHEMBL36535)
Affinity DataIC50: 43nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219797BDBM50219797(CHEMBL36934)
Affinity DataIC50: 46nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219796BDBM50219796(CHEMBL39464)
Affinity DataIC50: 50nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219800BDBM50219800(CHEMBL432475)
Affinity DataIC50: 83nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219806BDBM50219806(CHEMBL291140)
Affinity DataIC50: 94nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219809BDBM50219809(CHEMBL36643)
Affinity DataIC50: 110nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50102225BDBM50102225(N'-(3-[2,2']Bithiophenyl-5-yl-6,7-dichloro-quinoxa...)
Affinity DataIC50: 110nMAssay Description:Displacement of [125I]IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219811BDBM50219811(CHEMBL39710)
Affinity DataIC50: 160nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219812BDBM50219812(CHEMBL36842)
Affinity DataIC50: 200nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219794BDBM50219794(CHEMBL289656)
Affinity DataIC50: 220nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219808BDBM50219808(CHEMBL288527)
Affinity DataIC50: 220nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219810BDBM50219810(CHEMBL288876)
Affinity DataIC50: 360nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219795BDBM50219795(CHEMBL40080)
Affinity DataIC50: 410nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219789BDBM50219789(CHEMBL40955)
Affinity DataIC50: 680nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219793BDBM50219793(CHEMBL289789)
Affinity DataIC50: 760nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219790BDBM50219790(CHEMBL39937)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113636BDBM50113636([5-(4-Fluoro-phenylcarbamoyl)-pyridin-2-ylsulfanyl...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [125I]IL-8 from CHO cell membranes expressing human CX3C chemokine receptor 2 (CXCR2 filter mat binding assay)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219801BDBM50219801(CHEMBL40558)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219798BDBM50219798(CHEMBL39988)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219792BDBM50219792(CHEMBL40114)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219788BDBM50219788(CHEMBL36797)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219807BDBM50219807(CHEMBL288457)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50113636BDBM50113636([5-(4-Fluoro-phenylcarbamoyl)-pyridin-2-ylsulfanyl...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetC-X-C chemokine receptor type 1/2(Human)
Celltech R&D

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50219791BDBM50219791(CHEMBL35938)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition against GRO-alpha driven human neutrophil chemotaxisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed