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Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 50012035
TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataKi:  11nMAssay Description:Eq. constant (Ki) for inhibition of Cathepsin K was determined by progress curves, following hydrolysis of Z-Phe-Arg- Amc in the absence and presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataKi:  15nMAssay Description:Eq. constant (Ki) for inhibition of Cathepsin K was determined by progress curves, following hydrolysis of Z-Phe-Arg- Amc in the absence and presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113669(1-(2-Chloro-phenyl)-1H-[1,2,4]triazole-3-carboxyli...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  9nMAssay Description:Inhibition of recombinant human cathepsin K in fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113674(4-Methoxy-N-{(S)-1-[2-(4-methoxy-phenylamino)-ethy...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113673(4-Isopropyl-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  50nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113676((S)-benzyl 1-(2-(4-methoxyphenylamino)ethylamino)-...)
Affinity DataIC50:  60nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113665(CHEMBL308392 | [3-Methyl-1-(2-p-tolylamino-ethylca...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50:  190nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113668(CHEMBL78112 | {1-[2-(4-Chloro-phenylamino)-ethylca...)
Affinity DataIC50:  350nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113675(CHEMBL78288 | [3-Methyl-1-(2-m-tolylamino-ethylcar...)
Affinity DataIC50:  460nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113671(CHEMBL73908 | [3-Methyl-1-(2-phenylamino-ethylcarb...)
Affinity DataIC50:  470nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113666(CHEMBL78044 | {1-[2-(3-Methoxy-phenylamino)-ethylc...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin K(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113670(CHEMBL77335 | {1-[2-(3-Chloro-phenylamino)-ethylca...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of recombinant rabbit Cathepsin K in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113663(CHEMBL77471 | N-{1-[2-(4-Methoxy-phenylamino)-ethy...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113664(5-Isopropyl-pyridine-2-carboxylic acid {1-[2-(4-me...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113669(1-(2-Chloro-phenyl)-1H-[1,2,4]triazole-3-carboxyli...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113669(1-(2-Chloro-phenyl)-1H-[1,2,4]triazole-3-carboxyli...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113673(4-Isopropyl-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113664(5-Isopropyl-pyridine-2-carboxylic acid {1-[2-(4-me...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCathepsin S(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant human cathepsin S in a fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113662(1-(2,3-Dichloro-phenyl)-1H-[1,2,4]triazole-3-carbo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProcathepsin L(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50113667(4-Benzyloxy-N-{1-[2-(4-methoxy-phenylamino)-ethylc...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human cathepsin L in a fluorescence assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed