Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50037043
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115572BDBM50115572(CHEMBL18927 | CHEMBL492770 | 4-(3-Benzyloxy-phenyl...)
Affinity DataIC50: 350nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 107681BDBM107681(CHEMBL320261 | CHEMBL19977 | (2Z)-4-[3,5-bis(benzy...)
Affinity DataIC50: 480nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 107693BDBM107693(CHEMBL108760 | (2Z)-4-(5-chloro-1H-indol-3-yl)-2-h...)
Affinity DataIC50: 520nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093435BDBM50093435(1-(5-Chloro-1H-indol-3-yl)-3-hydroxy-3-(2H-tetrazo...)
Affinity DataIC50: 650nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370120BDBM50370120(CHEMBL611459)
Affinity DataIC50: 810nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115582BDBM50115582(4-[4-(3-Carboxy-3-hydroxy-acryloyl)-phenyl]-2-hydr...)
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115570BDBM50115570((Z)-2-Hydroxy-4-(1H-indol-3-yl)-4-oxo-but-2-enoic ...)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115575BDBM50115575(1-(5-Fluoro-1H-indol-3-yl)-3-hydroxy-3-(1H-tetrazo...)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115580BDBM50115580((Z)-4-[3-(3-Carboxy-3-hydroxy-acryloyl)-phenyl]-2-...)
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115573BDBM50115573(3-Hydroxy-1-(1H-indol-3-yl)-3-(1H-tetrazol-5-yl)-p...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115573BDBM50115573(3-Hydroxy-1-(1H-indol-3-yl)-3-(1H-tetrazol-5-yl)-p...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083953BDBM50083953((Z)-4-(3-Bromo-phenyl)-2-hydroxy-4-oxo-but-2-enoic...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083953BDBM50083953((Z)-4-(3-Bromo-phenyl)-2-hydroxy-4-oxo-but-2-enoic...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115588BDBM50115588(4-[2-(3-Carboxy-3-hydroxy-acryloyl)-quinolin-4-yl]...)
Affinity DataIC50: 6.50E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115587BDBM50115587(4-(5-Chloro-1H-indol-3-yl)-2-hydroxy-4-oxo-but-2-e...)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115582BDBM50115582(4-[4-(3-Carboxy-3-hydroxy-acryloyl)-phenyl]-2-hydr...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115582BDBM50115582(4-[4-(3-Carboxy-3-hydroxy-acryloyl)-phenyl]-2-hydr...)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115580BDBM50115580((Z)-4-[3-(3-Carboxy-3-hydroxy-acryloyl)-phenyl]-2-...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115581BDBM50115581(CHEMBL108423 | CHEMBL185721 | (Z)-2-Hydroxy-4-oxo-...)
Affinity DataIC50: 7.80E+3nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50370120BDBM50370120(CHEMBL611459)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115581BDBM50115581(CHEMBL108423 | CHEMBL185721 | (Z)-2-Hydroxy-4-oxo-...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115579BDBM50115579(CHEMBL16326 | (Z)-2-hydroxy-4-oxo-4-phenyl-but-2-e...)
Affinity DataIC50: 2.42E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115579BDBM50115579(CHEMBL16326 | (Z)-2-hydroxy-4-oxo-4-phenyl-but-2-e...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115577BDBM50115577(1-(5-Chloro-1H-indol-3-yl)-3-hydroxy-3-[1-(4-metho...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115574BDBM50115574(CHEMBL366966 | 4-(3-Benzoylamino-phenyl)-2-hydroxy...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093435BDBM50093435(1-(5-Chloro-1H-indol-3-yl)-3-hydroxy-3-(2H-tetrazo...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115586BDBM50115586(3-[3-Hydroxy-3-(1H-tetrazol-5-yl)-acryloyl]-1H-ind...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115586BDBM50115586(3-[3-Hydroxy-3-(1H-tetrazol-5-yl)-acryloyl]-1H-ind...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115572BDBM50115572(CHEMBL18927 | CHEMBL492770 | 4-(3-Benzyloxy-phenyl...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assay in experiment 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 107693BDBM107693(CHEMBL108760 | (2Z)-4-(5-chloro-1H-indol-3-yl)-2-h...)
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115575BDBM50115575(1-(5-Fluoro-1H-indol-3-yl)-3-hydroxy-3-(1H-tetrazo...)
Affinity DataIC50: 7.90E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115588BDBM50115588(4-[2-(3-Carboxy-3-hydroxy-acryloyl)-quinolin-4-yl]...)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115579BDBM50115579(CHEMBL16326 | (Z)-2-hydroxy-4-oxo-4-phenyl-but-2-e...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115574BDBM50115574(CHEMBL366966 | 4-(3-Benzoylamino-phenyl)-2-hydroxy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115576BDBM50115576(1-(3,5-Bis-benzyloxy-phenyl)-3-hydroxy-3-[1-(4-met...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115570BDBM50115570((Z)-2-Hydroxy-4-(1H-indol-3-yl)-4-oxo-but-2-enoic ...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115577BDBM50115577(1-(5-Chloro-1H-indol-3-yl)-3-hydroxy-3-[1-(4-metho...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115571BDBM50115571(3-[1-(3,5-Dimethoxy-benzyl)-1H-tetrazol-5-yl]-3-hy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115572BDBM50115572(CHEMBL18927 | CHEMBL492770 | 4-(3-Benzyloxy-phenyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assay in experiment 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115583BDBM50115583(3-Hydroxy-1-(1H-indol-3-yl)-3-[1-(4-methoxy-benzyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115585BDBM50115585((Z)-2-Hydroxy-4-oxo-4-quinolin-4-yl-but-2-enoic ac...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115581BDBM50115581(CHEMBL108423 | CHEMBL185721 | (Z)-2-Hydroxy-4-oxo-...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115576BDBM50115576(1-(3,5-Bis-benzyloxy-phenyl)-3-hydroxy-3-[1-(4-met...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115571BDBM50115571(3-[1-(3,5-Dimethoxy-benzyl)-1H-tetrazol-5-yl]-3-hy...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115585BDBM50115585((Z)-2-Hydroxy-4-oxo-4-quinolin-4-yl-but-2-enoic ac...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on strand transfer of proximal DNA into host DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115573BDBM50115573(3-Hydroxy-1-(1H-indol-3-yl)-3-(1H-tetrazol-5-yl)-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50083953BDBM50083953((Z)-4-(3-Bromo-phenyl)-2-hydroxy-4-oxo-but-2-enoic...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115587BDBM50115587(4-(5-Chloro-1H-indol-3-yl)-2-hydroxy-4-oxo-but-2-e...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50115583BDBM50115583(3-Hydroxy-1-(1H-indol-3-yl)-3-[1-(4-methoxy-benzyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
National Cancer Institute/Nih

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 107681BDBM107681(CHEMBL320261 | CHEMBL19977 | (2Z)-4-[3,5-bis(benzy...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory effect on 3'-processing(3'-P) of proximal DNA in an extracellular HIV-1 integrase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed