Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 50003619
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473868(CHEMBL339108)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473870(CHEMBL2112617)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473882(CHEMBL126206)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473876(CHEMBL2112614)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473868(CHEMBL339108)
Affinity DataKi:  60nMAssay Description:Displacement of verapamil from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473890(CHEMBL2111820)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473876(CHEMBL2112614)
Affinity DataIC50: 134nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473866(CHEMBL2112613)
Affinity DataKi:  149nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473883(CHEMBL2111817)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066066(CHEMBL281724 | (S)-1-[4-(Benzothiazol-2-yl-methyl-...)
Affinity DataKi:  203nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473881(CHEMBL2112615)
Affinity DataKi:  208nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473868(CHEMBL339108)
Affinity DataKi:  217nMAssay Description:Displacement of diltiazem from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473879(CHEMBL2111818)
Affinity DataKi:  241nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473882(CHEMBL126206)
Affinity DataIC50: 255nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473869(Lifarizine | RS-87476-000)
Affinity DataKi:  259nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473875(CHEMBL2111814)
Affinity DataKi:  312nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473870(CHEMBL2112617)
Affinity DataIC50: 322nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473868(CHEMBL339108)
Affinity DataIC50: 379nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473894(CHEMBL2112628)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473890(CHEMBL2111820)
Affinity DataKi:  391nMAssay Description:Displacement of diltiazem from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473870(CHEMBL2112617)
Affinity DataKi:  449nMAssay Description:Displacement of verapamil from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473883(CHEMBL2111817)
Affinity DataIC50: 452nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473869(Lifarizine | RS-87476-000)
Affinity DataIC50: 494nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473890(CHEMBL2111820)
Affinity DataKi:  500nMAssay Description:Displacement of verapamil from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473870(CHEMBL2112617)
Affinity DataKi:  660nMAssay Description:Displacement of diltiazem from L-type calcium channel binding siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473888(CHEMBL2111816)
Affinity DataKi:  662nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473891(CHEMBL2112624)
Affinity DataKi:  783nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473872(CHEMBL2111815)
Affinity DataKi:  864nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473890(CHEMBL2111820)
Affinity DataIC50: 922nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473881(CHEMBL2112615)
Affinity DataIC50: 975nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473880(CHEMBL421078)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473877(CHEMBL2111813)
Affinity DataKi:  1.23E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473887(CHEMBL2112616)
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473889(CHEMBL332216)
Affinity DataKi:  1.29E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473887(CHEMBL2112616)
Affinity DataKi:  1.33E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473879(CHEMBL2111818)
Affinity DataIC50: 1.48E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473886(CHEMBL2111819)
Affinity DataKi:  1.49E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473878(CHEMBL2112629)
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473885(CHEMBL2112618)
Affinity DataKi:  1.87E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473875(CHEMBL2111814)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473877(CHEMBL2111813)
Affinity DataIC50: 2.68E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066066(CHEMBL281724 | (S)-1-[4-(Benzothiazol-2-yl-methyl-...)
Affinity DataIC50: 2.94E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473880(CHEMBL421078)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473894(CHEMBL2112628)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473891(CHEMBL2112624)
Affinity DataIC50: 3.19E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473873(CHEMBL2111821)
Affinity DataKi:  3.31E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473886(CHEMBL2111819)
Affinity DataIC50: 3.77E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50066430(CHEMBL28854 | 2-(4-Methyl-piperazin-1-yl)-5-(2,3,5...)
Affinity DataKi:  4.00E+3nMAssay Description:Displacement of [3H]BTX from sodium channel of rat cerebral cortex synaptosomesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473873(CHEMBL2111821)
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rat)
Boehringer Ingelheim Pharma

Curated by ChEMBL
LigandPNGBDBM50473885(CHEMBL2112618)
Affinity DataIC50: 4.52E+3nMAssay Description:Inhibitory effect against veratridine-induced glutamate release from rat brain slicesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
Displayed 1 to 50 (of 77 total ) | Next | Last >>
Jump to: