Affinity DataKi: 5.10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.70nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 77nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 119nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 286nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKi: 1.73E+3nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataKd: 19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 1nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 7.94E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 3.98E+3nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 50.1nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 5.01E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 3.98E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: >3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 2.51E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 316nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 5.01E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 1.58E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 15.8nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin
Curated by ChEMBL
Freie Universit£T Berlin
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair