Compile Data Set for Download or QSAR
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Found 55 Enz. Inhib. hit(s) with all data for entry = 50037059
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118157(CHEMBL128635 | [1-(1-Methyl-cyclopropyl)-ethyl]-ca...)
Affinity DataKi:  5.10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118151(4-[3-(4,4-Dimethyl-pentyloxy)-propyl]-1H-imidazole...)
Affinity DataKi:  5.40nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118157(CHEMBL128635 | [1-(1-Methyl-cyclopropyl)-ethyl]-ca...)
Affinity DataKi:  6nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50370140(CHEMBL1788227)
Affinity DataKi:  6.70nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118159(CHEMBL340932 | Dicyclopropylmethyl-carbamic acid 3...)
Affinity DataKi:  8.20nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50370139(CHEMBL1788247)
Affinity DataKi:  9.70nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409581(CHEMBL2092970)
Affinity DataKi:  10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118156(4-[3-(3,3-Dimethyl-butoxy)-propyl]-1H-imidazole | ...)
Affinity DataKi:  10nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118156(4-[3-(3,3-Dimethyl-butoxy)-propyl]-1H-imidazole | ...)
Affinity DataKi:  11nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118159(CHEMBL340932 | Dicyclopropylmethyl-carbamic acid 3...)
Affinity DataKi:  11nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118155((1,2,2-Trimethyl-propyl)-carbamic acid 3-(1H-imida...)
Affinity DataKi:  13nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50370140(CHEMBL1788227)
Affinity DataKi:  13nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118152(4-[3-(5,5-Dimethyl-hexyloxy)-propyl]-1H-imidazole;...)
Affinity DataKi:  14nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118149((1-Cyclohexyl-ethyl)-carbamic acid 3-(1H-imidazol-...)
Affinity DataKi:  16nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118160((1-Cyclopropyl-ethyl)-carbamic acid 3-(1H-imidazol...)
Affinity DataKi:  20nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118162((Cyclopropyl-phenyl-methyl)-carbamic acid 3-(1H-im...)
Affinity DataKi:  44nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118153((Cyclohexyl-phenyl-methyl)-carbamic acid 3-(1H-imi...)
Affinity DataKi:  56nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118161((1-tert-Butyl-2,2-dimethyl-propyl)-carbamic acid 3...)
Affinity DataKi:  77nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118150(4-[3-(1,3,3-Trimethyl-butoxy)-propyl]-1H-imidazole...)
Affinity DataKi:  119nMAssay Description:In vitro inhibition of binding of [125I]iodoproxyfan against human Histamine H3 receptor stably transfected on CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118158(1-[3-(3,3-Dimethyl-butoxy)-propyl]-piperidine;1.1C...)
Affinity DataKi:  286nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118154(2,2-Dimethyl-propionic acid 3-(1H-imidazol-4-yl)-p...)
Affinity DataKi:  1.73E+3nMAssay Description:In vitro Histamine H3 receptor antagonist activity in synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118162((Cyclopropyl-phenyl-methyl)-carbamic acid 3-(1H-im...)
Affinity DataKd:  19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118159(CHEMBL340932 | Dicyclopropylmethyl-carbamic acid 3...)
Affinity DataKd:  1nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118161((1-tert-Butyl-2,2-dimethyl-propyl)-carbamic acid 3...)
Affinity DataKd:  1.26E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118162((Cyclopropyl-phenyl-methyl)-carbamic acid 3-(1H-im...)
Affinity DataKd:  3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118160((1-Cyclopropyl-ethyl)-carbamic acid 3-(1H-imidazol...)
Affinity DataKd:  2.00E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118153((Cyclohexyl-phenyl-methyl)-carbamic acid 3-(1H-imi...)
Affinity DataKd:  7.94E+3nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118160((1-Cyclopropyl-ethyl)-carbamic acid 3-(1H-imidazol...)
Affinity DataKd:  19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409579(CHEMBL130005)
Affinity DataKd:  3.98E+3nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118153((Cyclohexyl-phenyl-methyl)-carbamic acid 3-(1H-imi...)
Affinity DataKd:  100nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118150(4-[3-(1,3,3-Trimethyl-butoxy)-propyl]-1H-imidazole...)
Affinity DataKd:  50.1nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50370139(CHEMBL1788247)
Affinity DataKd:  5.01E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409580(CHEMBL131366)
Affinity DataKd:  19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409579(CHEMBL130005)
Affinity DataKd:  3.98E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118155((1,2,2-Trimethyl-propyl)-carbamic acid 3-(1H-imida...)
Affinity DataKd: >3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409580(CHEMBL131366)
Affinity DataKd: >1.00E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409578(CHEMBL2112321)
Affinity DataKd:  12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409579(CHEMBL130005)
Affinity DataKd:  3.16E+4nMAssay Description:Receptor profile was evaluated at Histamine H2 receptor of guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409578(CHEMBL2112321)
Affinity DataKd: >1.00E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118158(1-[3-(3,3-Dimethyl-butoxy)-propyl]-piperidine;1.1C...)
Affinity DataKd:  2.51E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118158(1-[3-(3,3-Dimethyl-butoxy)-propyl]-piperidine;1.1C...)
Affinity DataKd:  316nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50370139(CHEMBL1788247)
Affinity DataKd:  19.9nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118150(4-[3-(1,3,3-Trimethyl-butoxy)-propyl]-1H-imidazole...)
Affinity DataKd:  5.01E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118151(4-[3-(4,4-Dimethyl-pentyloxy)-propyl]-1H-imidazole...)
Affinity DataKd:  2.00E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118157(CHEMBL128635 | [1-(1-Methyl-cyclopropyl)-ethyl]-ca...)
Affinity DataKd:  1.58E+5nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118157(CHEMBL128635 | [1-(1-Methyl-cyclopropyl)-ethyl]-ca...)
Affinity DataKd:  15.8nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Cavia porcellus (domestic guinea pig))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118152(4-[3-(5,5-Dimethyl-hexyloxy)-propyl]-1H-imidazole;...)
Affinity DataKd:  1.00E+4nMAssay Description:Receptor profile was evaluated at Histamine H1 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118161((1-tert-Butyl-2,2-dimethyl-propyl)-carbamic acid 3...)
Affinity DataKd:  12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50409577(CHEMBL336499)
Affinity DataKd:  12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50118155((1,2,2-Trimethyl-propyl)-carbamic acid 3-(1H-imida...)
Affinity DataKd:  12.6nMAssay Description:Receptor profile was evaluated at Histamine H3 receptor of guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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