Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50012394
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118528BDBM50118528(Ethyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[e...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118528BDBM50118528(Ethyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[e...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118537BDBM50118537(Ethyl-carbamic acid 7-chloro-5-phenyl-6-oxa-10b-az...)
Affinity DataKi:  0.180nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118528BDBM50118528(Ethyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[e...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118539BDBM50118539(Diethyl-carbamic acid 5-thiophen-2-yl-6-oxa-10,10b...)
Affinity DataKi:  0.230nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118541BDBM50118541(Cyclopropyl-carbamic acid 5-phenyl-6-oxa-10b-aza-b...)
Affinity DataKi:  0.310nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118534BDBM50118534(Dimethyl-carbamic acid 5-p-tolyl-6-oxa-10,10b-diaz...)
Affinity DataKi:  0.440nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118541BDBM50118541(Cyclopropyl-carbamic acid 5-phenyl-6-oxa-10b-aza-b...)
Affinity DataKi:  0.470nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118542BDBM50118542(Diethyl-carbamic acid 5-m-tolyl-6-oxa-10,10b-diaza...)
Affinity DataKi:  0.560nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118545BDBM50118545(Ethyl-carbamic acid 5-p-tolyl-6-oxa-10b-aza-benzo[...)
Affinity DataKi:  0.680nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118544BDBM50118544(Methyl-propyl-carbamic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  0.690nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118527BDBM50118527(Methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[...)
Affinity DataKi:  0.760nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118543BDBM50118543(Ethyl-methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-...)
Affinity DataKi:  0.780nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118535BDBM50118535(Propyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[...)
Affinity DataKi:  0.910nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118529BDBM50118529(Butyl-methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118527BDBM50118527(Methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[...)
Affinity DataKi:  0.960nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118546BDBM50118546(Diethyl-carbamic acid 5-m-tolyl-6-oxa-10b-aza-benz...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118547BDBM50118547(Diethyl-carbamic acid 5-(3,5-difluoro-phenyl)-6-ox...)
Affinity DataKi:  1.26nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118531BDBM50118531(Diethyl-carbamic acid 5-phenyl-6-oxa-10,10b-diaza-...)
Affinity DataKi:  1.77nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118541BDBM50118541(Cyclopropyl-carbamic acid 5-phenyl-6-oxa-10b-aza-b...)
Affinity DataKi:  2.21nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118527BDBM50118527(Methyl-carbamic acid 5-phenyl-6-oxa-10b-aza-benzo[...)
Affinity DataKi:  2.26nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118540BDBM50118540(Acetic acid 5-m-tolyl-6-oxa-10b-aza-benzo[e]azulen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118530BDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118533BDBM50118533(Diethyl-carbamic acid 5-phenyl-6H-benzo[f]pyrrolo[...)
Affinity DataKi:  5.70nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118530BDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  6nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118530BDBM50118530(Azetidine-1-carboxylic acid 5-phenyl-6-oxa-10b-aza...)
Affinity DataKi:  6.03nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118536BDBM50118536(4-Methyl-piperazine-1-carboxylic acid 5-phenyl-6-o...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118531BDBM50118531(Diethyl-carbamic acid 5-phenyl-6-oxa-10,10b-diaza-...)
Affinity DataKi:  11nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118538BDBM50118538(Diethyl-carbamic acid 5-thiophen-2-yl-6-oxa-10b-az...)
Affinity DataKi:  11.5nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118532BDBM50118532(Acetic acid 5-p-tolyl-6-oxa-10,10b-diaza-benzo[e]a...)
Affinity DataKi:  13.5nMAssay Description:Inhibition of [3H]PK11195 binding to Peripheral type benzodiazepine receptor (PBR) in rat cortex homogenate by 50%More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118536BDBM50118536(4-Methyl-piperazine-1-carboxylic acid 5-phenyl-6-o...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118531BDBM50118531(Diethyl-carbamic acid 5-phenyl-6-oxa-10,10b-diaza-...)
Affinity DataKi:  22nMAssay Description:Inhibition of [3H]Ro-5-4864 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTranslocator protein(Rat)
Universita' Degli Studi Di Siena

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50118536BDBM50118536(4-Methyl-piperazine-1-carboxylic acid 5-phenyl-6-o...)
Affinity DataKi:  29nMAssay Description:Inhibition of [3H]PK11195 binding to mitochondrial rat testis Peripheral type benzodiazepine receptor (PBR)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed