Affinity DataKi: 26nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor at high affinity state expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.28E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.35E+4nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.36E+4nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor at low affinity state expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.10E+4nMAssay Description:Displacement [3H]DPCPX from of human adenosine A1 receptor expressed in CHO cells in presence of GTPMore data for this Ligand-Target Pair
Affinity DataKi: 3.25E+4nMAssay Description:Displacement of [3H]MSX-2 from A2A receptor in rat brain striatal membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Antagonist activity at adenosine A1 receptor in rat cortical membrane assessed as reduction of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 3.98E+3nMAssay Description:Agonist activity at adenosine A1 receptor in rat cortical membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 16.9nMAssay Description:Agonist activity at adenosine A1 receptor in rat cortical membrane by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair