Compile Data Set for Download or QSAR
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Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50037093
TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  0.100nMAssay Description:Binding affinity for opioid receptor like type, human Opioid receptor like 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  8.20nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  34nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  35nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  44nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  53nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  75nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  78nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  102nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  190nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121316(Ac-Arg-D-Cha-BTD-D-Arg-D-pClPhe-NH2 | CHEMBL358403)
Affinity DataKi:  222nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  270nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor mu 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  441nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  496nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  1.06E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  1.09E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  1.50E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor kappa 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  1.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  2.13E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121314(Ac-Arg-D-Cha-Phe-5-tBuPro-D-Arg-D-pClPhe-NH2 | CHE...)
Affinity DataKi:  2.34E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  2.70E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataKi:  5.20E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataKi:  7.05E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50094634(CHEMBL140979 | N-(4-Amino-2-methyl-quinolin-6-yl)-...)
Affinity DataKi:  8.65E+3nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121315(Ac-Arg-D-Cha-I9aa-D-Arg-D-pClPhe-NH2 | CHEMBL35621...)
Affinity DataKi:  1.09E+4nMAssay Description:Binding affinity for opioid receptor type, human Opioid receptor delta 1 expressed in membrane homogenates of COS-1 or CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataEC50:  1.40E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataEC50:  2.80E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor mu 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNociceptin receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50004178(Nociceptin | Nociceptin/orphanin FQ | ORPHANIN FQ)
Affinity DataEC50:  24nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding against human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121313(Ac-Arg-D-Cha-Qaa-D-Arg-D-pClPhe-NH2 | CHEMBL355931)
Affinity DataEC50: >1.00E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
University of Montreal

Curated by ChEMBL
LigandPNGBDBM50121312(Ac-Arg-D-Cha-I2aa-D-Arg-D-pClPhe-NH2 | CHEMBL26660...)
Affinity DataEC50: >1.00E+3nMAssay Description:Stimulation of [35S]GTP-gamma-S, binding using COS-human Opioid receptor kappa 1 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed