Affinity DataKi: 0.0210nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0350nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0420nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0470nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0630nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.233nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.241nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.289nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.301nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.411nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.443nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 1.22nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 5.49nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 6.92nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 21.7nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 47.1nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 47.5nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 53.9nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 80.3nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 272nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+3nMAssay Description:Inhibition of [3H]DAGO binding to Opioid receptor mu 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0150nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0260nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0350nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.120nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 1.21nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 6.36nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 16.5nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 40.7nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 71.7nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 108nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: >1.20E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 1.72E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 3.19E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 4.74E+3nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of guinea pig ileum (GPI)More data for this Ligand-Target Pair