Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50012741
LigandChemical structure of BindingDB Monomer ID 50122243BDBM50122243(4-chloro-5-(4-(furan-2-carbonyl)piperazin-1-yl)-2-...)
Affinity DataKi:  0.0520nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122242BDBM50122242(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortex using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122238BDBM50122238(4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-...)
Affinity DataKi:  0.220nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortex using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 29568BDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122239BDBM50122239(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122238BDBM50122238(4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222045BDBM50222045(CHEMBL45726)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122242BDBM50122242(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122243BDBM50122243(4-chloro-5-(4-(furan-2-carbonyl)piperazin-1-yl)-2-...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222044BDBM50222044(CHEMBL300092)
Affinity DataKi:  0.580nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122243BDBM50122243(4-chloro-5-(4-(furan-2-carbonyl)piperazin-1-yl)-2-...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortex using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50122239BDBM50122239(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222012BDBM50222012(CHEMBL49152)
Affinity DataKi:  1.40nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122242BDBM50122242(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222046BDBM50222046(CHEMBL46172)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat cerebral cortex using [3H]prazosinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122238BDBM50122238(4-chloro-5-(4-(2-(2-ethoxyphenoxy)ethyl)piperazin-...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 21393BDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50122239BDBM50122239(4-Chloro-5-{4-[2-(2-ethoxy-phenoxy)-ethyl]-piperaz...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50026636BDBM50026636(RAUWOLSCINE HYDROCHLORIDE | 17alpha-hydroxy-20alph...)
Affinity DataKi:  4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222045BDBM50222045(CHEMBL45726)
Affinity DataKi:  4nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222012BDBM50222012(CHEMBL49152)
Affinity DataKi:  4.60nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222044BDBM50222044(CHEMBL300092)
Affinity DataKi:  8.20nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50222046BDBM50222046(CHEMBL46172)
Affinity DataKi:  520nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor in rat cerebral cortex using [3H]rauwolscineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed