Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50012878
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123720(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50073047(CHEMBL291666 | N-[5-(3,4-Dimethoxy-phenyl)-1H-pyra...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123729(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  10nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50409778(CHEMBL2110162)
Affinity DataKi:  16nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123735(CHEMBL160443 | Indan-2-carboxylic acid [5-(3,4-dim...)
Affinity DataKi:  33nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123717(CHEMBL435036 | Indan-2-carboxylic acid [5-(4-chlor...)
Affinity DataKi:  59nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123726(CHEMBL159070 | Indan-2-carboxylic acid [5-(4-metho...)
Affinity DataKi:  62nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123727(CHEMBL158759 | Indan-2-carboxylic acid (5-p-tolyl-...)
Affinity DataKi:  80nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123728(CHEMBL160722 | Indan-2-carboxylic acid [5-(4-isopr...)
Affinity DataKi:  92nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123734(CHEMBL158940 | Indan-2-carboxylic acid [5-(3-chlor...)
Affinity DataKi:  120nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123732(CHEMBL161398 | Indan-2-carboxylic acid (5-phenyl-1...)
Affinity DataKi:  260nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123730(CHEMBL157588 | Indan-2-carboxylic acid [5-(2-chlor...)
Affinity DataKi:  450nMAssay Description:Inhibition of [125I]-PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataIC50:  14nMAssay Description:Antagonistic activity of compound was determined by its ability to inhibit NPY induced [Ca2+]i increases in CHO cells which expressed the recombinant...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataIC50:  14nMAssay Description:Antagonistic activity of compound was determined by its ability to inhibit NPY induced [Ca2+]i increases in CHO cells which expressed the recombinant...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50409778(CHEMBL2110162)
Affinity DataIC50:  16.3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123721(CHEMBL158732 | N-[5-(4-Chloro-phenyl)-1H-pyrazol-3...)
Affinity DataIC50:  47nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123723(CHEMBL160595 | N-[5-(4-Chloro-phenyl)-2H-pyrazol-3...)
Affinity DataIC50:  317nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123718(CHEMBL160389 | N-[5-(4-Chloro-phenyl)-2H-pyrazol-3...)
Affinity DataIC50:  443nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123719(CHEMBL350463 | N-[5-(4-Chloro-phenyl)-2H-pyrazol-3...)
Affinity DataIC50:  803nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123731(CHEMBL159134 | N-[5-(4-Chloro-phenyl)-2H-pyrazol-3...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123722(CHEMBL422185 | Naphthalene-2-carboxylic acid [5-(4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123733(CHEMBL158668 | Naphthalene-1-carboxylic acid [5-(4...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123736(Biphenyl-4-carboxylic acid [5-(4-chloro-phenyl)-2H...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 5(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123725(CHEMBL346300 | N-[5-(4-Chloro-phenyl)-2H-pyrazol-3...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of [125I]-PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed