Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50012878 Sort by
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataIC50: 14nMAssay Description:Antagonistic activity of compound was determined by its ability to inhibit NPY induced [Ca2+]i increases in CHO cells which expressed the recombinant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataIC50: 14nMAssay Description:Antagonistic activity of compound was determined by its ability to inhibit NPY induced [Ca2+]i increases in CHO cells which expressed the recombinant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50409778(CHEMBL2110162)
Affinity DataIC50: 16.3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123721(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-naphthal...)
Affinity DataIC50: 47nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123723(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-naphthal...)
Affinity DataIC50: 317nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123718(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-4-phenyl-b...)
Affinity DataIC50: 443nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123719(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-2-phenyl-a...)
Affinity DataIC50: 803nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123725(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-3-phenyl-p...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123736(Biphenyl-4-carboxylic acid [5-(4-chloro-phenyl)-2H...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123722(Naphthalene-2-carboxylic acid [5-(4-chloro-phenyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123733(Naphthalene-1-carboxylic acid [5-(4-chloro-phenyl)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123731(N-[5-(4-Chloro-phenyl)-2H-pyrazol-3-yl]-benzamide ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125I]PYY binding human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123720(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  2.80nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123724(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  7.30nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50073047(N-[5-(3,4-Dimethoxy-phenyl)-1H-pyrazol-3-yl]-2-nap...)
Affinity DataKi:  8.30nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123729(2,3-Dihydro-1H-cyclopenta[a]naphthalene-2-carboxyl...)
Affinity DataKi:  10nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50409778(CHEMBL2110162)
Affinity DataKi:  16nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123735(Indan-2-carboxylic acid [5-(3,4-dimethoxy-phenyl)-...)
Affinity DataKi:  33nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123717(N-(3-(4-chlorophenyl)-1H-pyrazol-5-yl)-2,3-dihydro...)
Affinity DataKi:  59nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123726(Indan-2-carboxylic acid [5-(4-methoxy-phenyl)-1H-p...)
Affinity DataKi:  62nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123727(Indan-2-carboxylic acid (5-p-tolyl-1H-pyrazol-3-yl...)
Affinity DataKi:  80nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123728(Indan-2-carboxylic acid [5-(4-isopropoxy-phenyl)-1...)
Affinity DataKi:  92nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123734(Indan-2-carboxylic acid [5-(3-chloro-phenyl)-1H-py...)
Affinity DataKi:  120nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123732(Indan-2-carboxylic acid (5-phenyl-1H-pyrazol-3-yl)...)
Affinity DataKi:  260nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuropeptide Y receptor type 5(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50123730(Indan-2-carboxylic acid [5-(2-chloro-phenyl)-1H-py...)
Affinity DataKi:  450nMAssay Description:Inhibition of [125I]PYY binding to human recombinant Neuropeptide Y receptor type 5 in LMtk-cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed