Compile Data Set for Download or QSAR
maximum 50k data
Found 49 Enz. Inhib. hit(s) with all data for entry = 50037232
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123752((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123763((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123756((E)-(1S,2R,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123754((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123750((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.290nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123751((E)-(1S,2S,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123759((E)-(1S,2S,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123762((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.440nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123760((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-etho...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123757((E)-(1S,2S,6R,7S)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123755(2-{(R)-2-[1-((S)-(S)-1-Carbamoyl-2-phenyl-ethylcar...)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123761((E)-(1S,2R,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123753((E)-(1S,2S,6R,7S)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123758((E)-(1S,2R,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123749((E)-(1S,2R,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DAMGO from human Opioid receptor mu 1 expressing CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123758((E)-(1S,2R,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  15nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123762((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123760((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-etho...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123759((E)-(1S,2S,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  21nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123763((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  22nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123749((E)-(1S,2R,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  25nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123751((E)-(1S,2S,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123759((E)-(1S,2S,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123763((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123750((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  42nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123758((E)-(1S,2R,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123753((E)-(1S,2S,6R,7S)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  50nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123756((E)-(1S,2R,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  51nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123752((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123754((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123757((E)-(1S,2S,6R,7S)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  60nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123751((E)-(1S,2S,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  64nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123761((E)-(1S,2R,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123761((E)-(1S,2R,6R,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  69nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123752((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  69nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123749((E)-(1S,2R,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123762((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  85nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123750((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  99nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123757((E)-(1S,2S,6R,7S)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123756((E)-(1S,2R,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  123nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123760((E)-(1S,2S,6S,7R)-7-((S)-1-Carbamoyl-2-phenyl-etho...)
Affinity DataKi:  126nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123753((E)-(1S,2S,6R,7S)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123754((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataKi:  260nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123755(2-{(R)-2-[1-((S)-(S)-1-Carbamoyl-2-phenyl-ethylcar...)
Affinity DataKi:  1.04E+4nMAssay Description:Displacement of 3H-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellum preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123755(2-{(R)-2-[1-((S)-(S)-1-Carbamoyl-2-phenyl-ethylcar...)
Affinity DataKi:  2.50E+4nMAssay Description:Displacement of [3H]diprenorphine from human Opioid receptor delta 1 epressing HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123755(2-{(R)-2-[1-((S)-(S)-1-Carbamoyl-2-phenyl-ethylcar...)
Affinity DataEC50:  31nMAssay Description:Compound tested at 10 uM for the ability to induce Opioid receptor mu 1-mediated binding of [35S]GTP-gamma-S to G proteins in CHO membrane preparatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123759((E)-(1S,2S,6R,7R)-7-((S)-1-Carbamoyl-2-phenyl-ethy...)
Affinity DataEC50:  7.90nMAssay Description:Compound tested at 10 uM for the ability to induce Opioid receptor mu 1-mediated binding of [35S]GTP-gamma-S to G proteins in CHO membrane preparatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123756((E)-(1S,2R,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataEC50:  49nMAssay Description:Compound tested at 10 uM for the ability to induce Opioid receptor mu 1-mediated binding of [35S]GTP-gamma-S to G proteins in CHO membrane preparatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Harvard University

Curated by ChEMBL
LigandPNGBDBM50123754((E)-(1S,2S,6S,7R)-2,6-Dihydroxy-1-(4-hydroxy-2,6-d...)
Affinity DataEC50:  4.20nMAssay Description:Compound tested at 10 uM for the ability to induce Opioid receptor mu 1-mediated binding of [35S]GTP-gamma-S to G proteins in CHO membrane preparatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed