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Found 19 Enz. Inhib. hit(s) with all data for entry = 50012980
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124971((2R,3S)-5,6,8,5',6',8'-Hexahydroxy-2,3,2',3'-tetra...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124967(5,6,8,5',6',8'-Hexahydroxy-2,3,2',3'-tetramethyl-2...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124967(5,6,8,5',6',8'-Hexahydroxy-2,3,2',3'-tetramethyl-2...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124966((8R,9R)-2,4,5-Trihydroxy-8,9-dimethyl-1-((2S,3R)-5...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124971((2R,3S)-5,6,8,5',6',8'-Hexahydroxy-2,3,2',3'-tetra...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124964(6,8'-Dihydroxy-5,8,5',6'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124966((8R,9R)-2,4,5-Trihydroxy-8,9-dimethyl-1-((2S,3R)-5...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124967(5,6,8,5',6',8'-Hexahydroxy-2,3,2',3'-tetramethyl-2...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124970(6-Hydroxy-5,8,5',6',8'-pentamethoxy-2,3,2',3'-tetr...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124968(Acetic acid 6,8,5',6',8'-pentaacetoxy-2,3,2',3'-te...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124969(5,6,8,5',6',8'-Hexamethoxy-2,3,2',3'-tetramethyl-2...)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124965(5,6-Dihydroxy-8,5',6',8'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124965(5,6-Dihydroxy-8,5',6',8'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50:  8.00E+4nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124965(5,6-Dihydroxy-8,5',6',8'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124968(Acetic acid 6,8,5',6',8'-pentaacetoxy-2,3,2',3'-te...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124964(6,8'-Dihydroxy-5,8,5',6'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124965(5,6-Dihydroxy-8,5',6',8'-tetramethoxy-2,3,2',3'-te...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124969(5,6,8,5',6',8'-Hexamethoxy-2,3,2',3'-tetramethyl-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in coupled transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124970(6-Hydroxy-5,8,5',6',8'-pentamethoxy-2,3,2',3'-tetr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of HIV-1 integrase in strand transfer assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed