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Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50041068
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.180nMAssay Description:In vitro inhibitory potency for preventing ET-1 induced constriction of rat aortic rings (ETA receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50125187(2-(2-Chloro-pyrimidin-5-yl)-7-aza-bicyclo[2.2.1]he...)
Affinity DataKi:  0.310nMAssay Description:In vitro inhibitory potency for preventing sarafotoxin S6c induced constriction of rat tracheal rings (ETB receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50125188(CHEMBL268176 | N-[5-(7-Aza-bicyclo[2.2.1]hept-2-yl...)
Affinity DataKi:  16nMAssay Description:In vitro inhibitory potency for preventing ET-1 induced constriction of rat aortic rings (ETA receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Louis Pasteur University

Curated by ChEMBL
LigandPNGBDBM50125189(CHEMBL267191 | [5-(7-Aza-bicyclo[2.2.1]hept-2-yl)-...)
Affinity DataKi:  8.10E+3nMAssay Description:In vitro inhibitory potency for preventing ET-1 induced constriction of rat aortic rings (ETA receptor)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed