Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50013078
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126193BDBM50126193({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126188BDBM50126188([4-(9-Propylcarbamoyl-9H-fluoren-9-yl)-butyl]-phos...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126207BDBM50126207((4-{9-[2-(4-Methoxy-phenyl)-ethylcarbamoyl]-9H-flu...)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126201BDBM50126201({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126201BDBM50126201({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126209BDBM50126209({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126225BDBM50126225({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126212BDBM50126212({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 27nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126223BDBM50126223({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126192BDBM50126192({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126222BDBM50126222({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126189BDBM50126189({6-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 45nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126198BDBM50126198({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 55nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126194BDBM50126194({5-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126211BDBM50126211({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 85nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126220BDBM50126220({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 90nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126216BDBM50126216([4-(9-Propylcarbamoyl-9H-fluoren-9-yl)-butyl]-phos...)
Affinity DataIC50: 135nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126217BDBM50126217({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 145nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126200BDBM50126200(9-[3-(4-Benzoylamino-piperidin-1-yl)-propyl]-9H-fl...)
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126187BDBM50126187([4-(9-Benzylcarbamoyl-9H-fluoren-9-yl)-butyl]-phos...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126214BDBM50126214({4-[9-(2,2,2-Trifluoro-ethylcarbamoyl)-9H-fluoren-...)
Affinity DataIC50: 280nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126203BDBM50126203([4-(9-Butylcarbamoyl-9H-fluoren-9-yl)-butyl]-phosp...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126206BDBM50126206(9-[4-(Dibutoxy-phosphoryl)-butyl]-9H-fluorene-9-ca...)
Affinity DataIC50: 450nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126224BDBM50126224((4-{9-[(Pyridin-2-ylmethyl)-carbamoyl]-9H-fluoren-...)
Affinity DataIC50: 470nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126197BDBM50126197({4-[9-(2-Morpholin-4-yl-ethylcarbamoyl)-9H-fluoren...)
Affinity DataIC50: 500nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126210BDBM50126210({4-[9-(4-Amino-benzylcarbamoyl)-9H-fluoren-9-yl]-b...)
Affinity DataIC50: 890nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126204BDBM50126204(2-[1-(3,3-Diphenyl-propyl)-piperidin-4-yl]-2,3-dih...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126202BDBM50126202(9-Allyl-9H-fluorene-9-carboxylic acid ethylamide |...)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126205BDBM50126205([3-(6-Ethoxy-benzothiazol-2-ylsulfanyl)-propyl]-ph...)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126195BDBM50126195((3-Phenoxy-propyl)-phosphonic acid dibutyl ester |...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126218BDBM50126218([3-(6-Ethoxy-benzooxazol-2-ylsulfanyl)-propyl]-pho...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126221BDBM50126221([3-(6-Ethoxy-1-methyl-1H-benzoimidazol-2-ylsulfany...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126199BDBM50126199([5-(6-Ethoxy-benzothiazol-2-ylsulfanyl)-pentyl]-ph...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126196BDBM50126196([3-(4,5-Diphenyl-oxazol-2-ylsulfanyl)-propyl]-phos...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126190BDBM50126190([3-(6-Ethoxy-1H-benzoimidazol-2-ylsulfanyl)-propyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126191BDBM50126191([4-(6-Ethoxy-benzothiazol-2-ylsulfanyl)-butyl]-pho...)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126215BDBM50126215([3-(Pyridin-4-ylsulfanyl)-propyl]-phosphonic acid ...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126219BDBM50126219([3-(Naphthalen-1-yloxy)-propyl]-phosphonic acid di...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126213BDBM50126213([3-(4,5-Diphenyl-1H-imidazol-2-ylsulfanyl)-propyl]...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMicrosomal triglyceride transfer protein large subunit(Bovine)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50126208BDBM50126208([3-(Thiophen-2-ylsulfanyl)-propyl]-phosphonic acid...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against microsomal triglyceride transfer protein (MTP)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed