Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50013083
LigandPNGBDBM50126336(4-{[(4-Cyano-3-naphthalen-1-yl-phenyl)-(3-methyl-3...)
Affinity DataIC50:  0.370nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126339(4-[(3-CYANO-BENZYL)-(3-METHYL-3H-IMIDAZOL-4-YLMETH...)
Affinity DataIC50:  0.390nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
LigandPNGBDBM50126340(4-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  0.450nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126335(6-[(R)-Amino-(4-chloro-phenyl)-(3-methyl-3H-imidaz...)
Affinity DataIC50:  0.570nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB

LigandPNGBDBM50126330(5-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  0.970nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM17325((2S)-2-[(4-{[butyl(2-cyclohexylethyl)amino]methyl}...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
LigandPNGBDBM50126331(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126337(4-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126331(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126333(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50:  1.90nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM14459((+)-4-[2-[4-(8-Chloro-3,10-dibromo-6,11-dihydro-5H...)
Affinity DataIC50:  7.80nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
LigandPNGBDBM50126334(5-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  10nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126344(5-[Benzyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126329(CHEMBL28588 | N-(4-Cyano-3-naphthalen-1-yl-phenyl)...)
Affinity DataIC50:  14nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126338(CHEMBL28490 | N-(4-Cyano-3-naphthalen-1-yl-phenyl)...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126328(4-[(3-Methyl-3H-imidazol-4-ylmethyl)-amino]-2-naph...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126328(4-[(3-Methyl-3H-imidazol-4-ylmethyl)-amino]-2-naph...)
Affinity DataIC50:  31nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126341(4-[Methyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126341(4-[Methyl-(3-methyl-3H-imidazol-4-ylmethyl)-amino]...)
Affinity DataIC50:  38nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126343(5-[Benzyloxy-(3-methyl-3H-imidazol-4-yl)-methyl]-2...)
Affinity DataIC50:  65nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126332(5-[Benzyl-(3H-imidazol-4-ylmethyl)-amino]-2'-methy...)
Affinity DataIC50:  84nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126339(4-[(3-CYANO-BENZYL)-(3-METHYL-3H-IMIDAZOL-4-YLMETH...)
Affinity DataIC50:  150nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
LigandPNGBDBM50126333(4-[Cyclohexyl-(3-methyl-3H-imidazol-4-ylmethyl)-am...)
Affinity DataIC50:  180nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126340(4-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  230nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126329(CHEMBL28588 | N-(4-Cyano-3-naphthalen-1-yl-phenyl)...)
Affinity DataIC50:  310nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126336(4-{[(4-Cyano-3-naphthalen-1-yl-phenyl)-(3-methyl-3...)
Affinity DataIC50:  650nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126337(4-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibition of geranylgeranyltransferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126334(5-[(4-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126342(2'-Methyl-5-[(3-methyl-3H-imidazol-4-ylmethyl)-ami...)
Affinity DataIC50:  1.00E+3nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126330(5-[(3-Cyano-benzyl)-(3-methyl-3H-imidazol-4-ylmeth...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50126338(CHEMBL28490 | N-(4-Cyano-3-naphthalen-1-yl-phenyl)...)
Affinity DataIC50:  1.90E+3nMAssay Description:In vitro inhibitory activity of the compound against farnesyltransferase (FTase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed