Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50013105 Sort by
TargetKappa-type opioid receptor(Guinea pig)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(Compound [Gly2]Venorphin | CHEMBL263595)
Affinity DataKi:  8.40nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in Chinese hamster ovary cells expressing cloned opioid recep...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(Compound Venorphin | CHEMBL438571)
Affinity DataKi:  20nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in Chinese hamster ovary cells expressing cloned opioid recep...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-Arg-Ile-Arg-Pro-...)
Affinity DataKi:  27nMAssay Description:Binding affinity towards Opioid receptor kappa 1 using [3H]diprenorphine as radioligand in Chinese hamster ovary cells expressing cloned opioid recep...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(Compound Venorphin | CHEMBL438571)
Affinity DataKi:  251nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-Arg-Ile-Arg-Pro-...)
Affinity DataKi:  331nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMu-type opioid receptor(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(Compound [Gly2]Venorphin | CHEMBL263595)
Affinity DataKi:  339nMAssay Description:Binding affinity towards Opioid receptor mu 1 using [3H]DAMGO as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126658(Compound Venorphin | CHEMBL438571)
Affinity DataKi:  5.32E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126657(cyclo(1-5)Tyr-Gly-Trp-Trp-Glu-Arg-Arg-Ile-Arg-Pro-...)
Affinity DataKi: >8.90E+3nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50126656(Compound [Gly2]Venorphin | CHEMBL263595)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity towards Opioid receptor delta 1 using [3H]DPDPE as radioligand in Chinese hamster ovary cells expressing cloned opioid receptorsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed