Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50013151
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127191(2-(8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127179(2-{8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  4.20nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50116238(8-(2-Fluoro-benzyl)-2-(4-methoxy-phenyl)-6-(3-meth...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity to human Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127199(8-(2-fluorobenzyl)-2-tert-butyl-6-(3-methoxyphenyl...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127196(2-tert-Butyl-3-{[ethyl-(2-pyridin-2-yl-ethyl)-amin...)
Affinity DataKi:  7.90nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127195(8-(2-Fluoro-benzyl)-2-(2-hydroxy-1,1-dimethyl-ethy...)
Affinity DataKi:  8nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127187(2-tert-Butyl-8-(2-fluoro-benzyl)-6-(3-methoxy-phen...)
Affinity DataKi:  11nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127186(2-tert-Butyl-8-(2-fluoro-benzyl)-6-(3-methoxy-phen...)
Affinity DataKi:  30nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127190(2-[3-[(Benzyl-methyl-amino)-methyl]-8-(2-fluoro-be...)
Affinity DataKi:  59nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127180(3-[(Benzyl-methyl-amino)-methyl]-2-tert-butyl-8-(2...)
Affinity DataKi:  72nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127177(2-{8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  130nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127188(2-tert-Butyl-8-(2-fluoro-benzyl)-6-(3-methoxy-phen...)
Affinity DataKi:  160nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127192(2-tert-Butyl-8-(2-fluoro-benzyl)-6-(3-methoxy-phen...)
Affinity DataKi:  190nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127181(3-(Benzylamino-methyl)-2-tert-butyl-8-(2-fluoro-be...)
Affinity DataKi:  240nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127185(2-tert-Butyl-3-{[(2-diethylamino-ethyl)-methyl-ami...)
Affinity DataKi:  260nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127197(2-[8-(2-Fluoro-benzyl)-3-{[(2-methoxy-ethyl)-methy...)
Affinity DataKi:  300nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127189(2-[3-[(Butyl-methyl-amino)-methyl]-8-(2-fluoro-ben...)
Affinity DataKi:  320nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127200(2-[1,1-Dimethyl-2-(2-pyridin-2-yl-ethylamino)-ethy...)
Affinity DataKi:  350nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127201(2-{8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  400nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127193(2-tert-Butyl-8-(2-fluoro-benzyl)-3-{[(2-methoxy-et...)
Affinity DataKi:  430nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127194(2-tert-Butyl-3-[(cyclohexylmethyl-amino)-methyl]-8...)
Affinity DataKi:  430nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127198(2-[8-(2-Fluoro-benzyl)-3-{[(2-hydroxy-benzyl)-meth...)
Affinity DataKi:  490nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127184(2-tert-Butyl-3-dimethylaminomethyl-8-(2-fluoro-ben...)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127176(2-[8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127202(2-tert-Butyl-3-[(cyclopentylmethyl-amino)-methyl]-...)
Affinity DataKi:  6.40E+3nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127178(2-[8-(2-Fluoro-benzyl)-6-(3-methoxy-phenyl)-7-meth...)
Affinity DataKi:  7.70E+3nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127182(2-[3-(3,4-Dihydro-1H-isoquinolin-2-ylmethyl)-8-(2-...)
Affinity DataKi:  9.20E+3nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandPNGBDBM50127183(1-(2-Fluoro-benzyl)-3-(3-methoxy-phenyl)-2,8,8-tri...)
Affinity DataKi:  1.20E+4nMAssay Description:Binding affinity against human gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed