Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50013162
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50075009(1-Ethyl-5-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50: 41nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127282(7-[(4-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50: 55nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127279(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50: 62nMAssay Description:In vitro inhibition of cytochrome P450 19A1 from human placental microsomes with 2.5 uM [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127286(1-Ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl-methyl]...)
Affinity DataIC50: 62nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127285(5-Chloro-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-y...)
Affinity DataIC50: 63nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127281(7-[(4-Bromo-phenyl)-imidazol-1-yl-methyl]-1-ethyl-...)
Affinity DataIC50: 70nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127280(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50: 90nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127283(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50: 110nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127284(7-[(3-Chloro-phenyl)-imidazol-1-yl-methyl]-1-ethyl...)
Affinity DataIC50: 170nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127287(5-Bromo-1-ethyl-7-[(4-fluoro-phenyl)-imidazol-1-yl...)
Affinity DataIC50: 200nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM50127278(1-Ethyl-7-[(4-fluoro-phenyl)-[1,2,4]triazol-1-yl-m...)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAromatase(Human)
Ufr Des Sciences Pharmaceutiques

Curated by ChEMBL
LigandPNGBDBM9460(3-(4-aminophenyl)-3-ethyl-piperidine-2,6-dione | C...)
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of cytochrome P450 19A1 of human placental microsomes with [1-beta,2beta-3H]testosteroneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed